{"data":{"id":3999,"citation":"Khedkar NR, Irlapatti NR, Dadke D, Kanoje V, Shaikh Z, Karche V, Shinde V, Deshmukh G, Patil A, Jachak S, Phukan S, Kizhakinagath PA, Gholve M, Bhankhede T, Daler J, Nemade HN, Budhe S, Pareek H, Yeshodharan R, Gupta R, Kalia A, Pandey D, Wagh A, Kumar S, Patil V, Modi D, Sharma N, Ahirrao P, Mehta M, Kumar H, Nigade P, Tamane K, Mallurwar S, Kuldharan S, Pawar S, Vishwase G, Bokan S, Singh M, Naik K, Ingawale S, Shankar R, Kamalakannan P, Venugopal S, George SK, Padiya KJ, Nemmani KVS, Gundu J, Bhonde M, Narasimham L, Sindkhedkar M, Shah C, Sinha N, Sharma S, Bakhle D, Kamboj RK, Palle VP.: Discovery of a Novel Potent and Selective Calcium Release-Activated Calcium Channel Inhibitor: 2,6-Difluoro-<i>N<\/i>-(2'-methyl-3'-(4-methyl-5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)-[1,1'-biphenyl]-4-yl)benzamide. Structure-Activity Relationship and Preclinical Characterization. J Med Chem, Volume 64 (23), 2021","title":"Discovery of a Novel Potent and Selective Calcium Release-Activated Calcium Channel Inhibitor: 2,6-Difluoro-<i>N<\/i>-(2'-methyl-3'-(4-methyl-5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)-[1,1'-biphenyl]-4-yl)benzamide. Structure-Activity Relationship and Preclinical Characterization.","doi":"10.1021\/acs.jmedchem.1c01403","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.1c01403","pmid":"34843241","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/34843241\/","year":2021,"journal":"J Med Chem","volume":"64","issue":"23","page":"17004-17030","authors":[{"first_name":"Ahirrao P","last_name":null,"full_name":null},{"first_name":"Bhankhede T","last_name":null,"full_name":null},{"first_name":"Budhe S","last_name":null,"full_name":null},{"first_name":"Dadke D","last_name":null,"full_name":null},{"first_name":"Daler J","last_name":null,"full_name":null},{"first_name":"Deshmukh G","last_name":null,"full_name":null},{"first_name":"Gholve M","last_name":null,"full_name":null},{"first_name":"Gupta R","last_name":null,"full_name":null},{"first_name":"Irlapatti NR","last_name":null,"full_name":null},{"first_name":"Jachak S","last_name":null,"full_name":null},{"first_name":"Kalia A","last_name":null,"full_name":null},{"first_name":"Kanoje V","last_name":null,"full_name":null},{"first_name":"Karche V","last_name":null,"full_name":null},{"first_name":"Khedkar NR","last_name":null,"full_name":null},{"first_name":"Kizhakinagath PA","last_name":null,"full_name":null},{"first_name":"Kuldharan S","last_name":null,"full_name":null},{"first_name":"Kumar H","last_name":null,"full_name":null},{"first_name":"Kumar S","last_name":null,"full_name":null},{"first_name":"Mallurwar S","last_name":null,"full_name":null},{"first_name":"Mehta M","last_name":null,"full_name":null},{"first_name":"Modi D","last_name":null,"full_name":null},{"first_name":"Nemade HN","last_name":null,"full_name":null},{"first_name":"Nigade P","last_name":null,"full_name":null},{"first_name":"Pandey D","last_name":null,"full_name":null},{"first_name":"Pareek H","last_name":null,"full_name":null},{"first_name":"Patil A","last_name":null,"full_name":null},{"first_name":"Patil V","last_name":null,"full_name":null},{"first_name":"Phukan S","last_name":null,"full_name":null},{"first_name":"Shaikh Z","last_name":null,"full_name":null},{"first_name":"Sharma N","last_name":null,"full_name":null},{"first_name":"Shinde V","last_name":null,"full_name":null},{"first_name":"Tamane K","last_name":null,"full_name":null},{"first_name":"Wagh A","last_name":null,"full_name":null},{"first_name":"Yeshodharan R","last_name":null,"full_name":null},{"first_name":"Bakhle D","last_name":null,"full_name":null},{"first_name":"Bhonde M","last_name":null,"full_name":null},{"first_name":"Bokan S","last_name":null,"full_name":null},{"first_name":"George SK","last_name":null,"full_name":null},{"first_name":"Gundu J","last_name":null,"full_name":null},{"first_name":"Ingawale S","last_name":null,"full_name":null},{"first_name":"Kamalakannan P","last_name":null,"full_name":null},{"first_name":"Kamboj RK","last_name":null,"full_name":null},{"first_name":"Naik K","last_name":null,"full_name":null},{"first_name":"Narasimham L","last_name":null,"full_name":null},{"first_name":"Nemmani KVS","last_name":null,"full_name":null},{"first_name":"Padiya KJ","last_name":null,"full_name":null},{"first_name":"Palle VP.","last_name":null,"full_name":null},{"first_name":"Pawar S","last_name":null,"full_name":null},{"first_name":"Shah C","last_name":null,"full_name":null},{"first_name":"Shankar R","last_name":null,"full_name":null},{"first_name":"Sharma S","last_name":null,"full_name":null},{"first_name":"Sindkhedkar M","last_name":null,"full_name":null},{"first_name":"Singh M","last_name":null,"full_name":null},{"first_name":"Sinha N","last_name":null,"full_name":null},{"first_name":"Venugopal S","last_name":null,"full_name":null},{"first_name":"Vishwase G","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3999","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3999","created_at":"2024-05-21T20:14:30.000000Z","updated_at":null}}