{"data":{"id":3943,"citation":"Prime ME, Andersen OA, Barker JJ, Brooks MA, Cheng RK, Toogood-Johnson I, Courtney SM, Brookfield FA, Yarnold CJ, Marston RW, Johnson PD, Johnsen SF, Palfrey JJ, Vaidya D, Erfan S, Ichihara O, Felicetti B, Palan S, Pedret-Dunn A, Schaertl S, Sternberger I, Ebneth A, Scheel A, Winkler D, Toledo-Sherman L, Beconi M, Macdonald D, Mu\u00f1oz-Sanjuan I, Dominguez C, Wityak J.: Discovery and structure-activity relationship of potent and selective covalent inhibitors of transglutaminase 2 for Huntington's disease. J Med Chem, Volume 55 (3), 2012","title":"Discovery and structure-activity relationship of potent and selective covalent inhibitors of transglutaminase 2 for Huntington's disease.","doi":"10.1021\/jm201310y","doi_url":"https:\/\/doi.org\/10.1021\/jm201310y","pmid":"22224594","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/22224594\/","year":2012,"journal":"J Med Chem","volume":"55","issue":"3","page":"1021-1046","authors":[{"first_name":"Andersen OA","last_name":null,"full_name":null},{"first_name":"Barker JJ","last_name":null,"full_name":null},{"first_name":"Beconi M","last_name":null,"full_name":null},{"first_name":"Brookfield FA","last_name":null,"full_name":null},{"first_name":"Brooks MA","last_name":null,"full_name":null},{"first_name":"Cheng RK","last_name":null,"full_name":null},{"first_name":"Courtney SM","last_name":null,"full_name":null},{"first_name":"Dominguez C","last_name":null,"full_name":null},{"first_name":"Ebneth A","last_name":null,"full_name":null},{"first_name":"Erfan S","last_name":null,"full_name":null},{"first_name":"Felicetti B","last_name":null,"full_name":null},{"first_name":"Ichihara O","last_name":null,"full_name":null},{"first_name":"Johnsen SF","last_name":null,"full_name":null},{"first_name":"Johnson PD","last_name":null,"full_name":null},{"first_name":"MacDonald D","last_name":null,"full_name":null},{"first_name":"Marston RW","last_name":null,"full_name":null},{"first_name":"Munoz-Sanjuan I","last_name":null,"full_name":null},{"first_name":"Palan S","last_name":null,"full_name":null},{"first_name":"Palfrey JJ","last_name":null,"full_name":null},{"first_name":"Pedret-Dunn A","last_name":null,"full_name":null},{"first_name":"Prime ME","last_name":null,"full_name":null},{"first_name":"Schaertl S","last_name":null,"full_name":null},{"first_name":"Scheel A","last_name":null,"full_name":null},{"first_name":"Sternberger I","last_name":null,"full_name":null},{"first_name":"Toledo-Sherman L","last_name":null,"full_name":null},{"first_name":"Toogood-Johnson I","last_name":null,"full_name":null},{"first_name":"Vaidya D","last_name":null,"full_name":null},{"first_name":"Winkler D","last_name":null,"full_name":null},{"first_name":"Wityak J.","last_name":null,"full_name":null},{"first_name":"Yarnold CJ","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3943","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3943","created_at":"2024-05-21T20:14:13.000000Z","updated_at":null}}