{"data":{"id":3894,"citation":"Wanner J, Chen L, Lemoine RC, Kondru R, Jekle A, Heilek G, deRosier A, Ji C, Berry PW, Rotstein DM.: Evaluation of amide replacements in CCR5 antagonists as a means to increase intrinsic permeability. Part 2: SAR optimization and pharmacokinetic profile of a homologous azacyle series. Bioorg Med Chem Lett, Volume 20 (22), 2010","title":"Evaluation of amide replacements in CCR5 antagonists as a means to increase intrinsic permeability. Part 2: SAR optimization and pharmacokinetic profile of a homologous azacyle series.","doi":"10.1016\/j.bmcl.2010.08.118","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2010.08.118","pmid":"20855212","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20855212\/","year":2010,"journal":"Bioorg Med Chem Lett","volume":"20","issue":"22","page":"6802-6807","authors":[{"first_name":"Berry PW","last_name":null,"full_name":null},{"first_name":"Chen L","last_name":null,"full_name":null},{"first_name":"deRosier A","last_name":null,"full_name":null},{"first_name":"Heilek G","last_name":null,"full_name":null},{"first_name":"Jekle A","last_name":null,"full_name":null},{"first_name":"Ji C","last_name":null,"full_name":null},{"first_name":"Kondru R","last_name":null,"full_name":null},{"first_name":"Lemoine RC","last_name":null,"full_name":null},{"first_name":"Rotstein DM.","last_name":null,"full_name":null},{"first_name":"Wanner J","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3894","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3894","created_at":"2024-05-21T20:14:01.000000Z","updated_at":null}}