{"data":{"id":3870,"citation":"D\u00edaz JL, Cuberes R, Berrocal J, Contijoch M, Christmann U, Fern\u00e1ndez A, Port A, Holenz J, Buschmann H, Laggner C, Serafini MT, Burgue\u00f1o J, Zamanillo D, Merlos M, Vela JM, Almansa C.: Synthesis and biological evaluation of the 1-arylpyrazole class of \u03c3(1) receptor antagonists: identification of 4-{2-[5-methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine (S1RA, E-52862). J Med Chem, Volume 55 (19), 2012","title":"Synthesis and biological evaluation of the 1-arylpyrazole class of \u03c3(1) receptor antagonists: identification of 4-{2-[5-methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine (S1RA, E-52862).","doi":"10.1021\/jm3007323","doi_url":"https:\/\/doi.org\/10.1021\/jm3007323","pmid":"22784008","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/22784008\/","year":2012,"journal":"J Med Chem","volume":"55","issue":"19","page":"8211-8224","authors":[{"first_name":"Berrocal J","last_name":null,"full_name":null},{"first_name":"Burgue\u00f1o J","last_name":null,"full_name":null},{"first_name":"Buschmann H","last_name":null,"full_name":null},{"first_name":"Christmann U","last_name":null,"full_name":null},{"first_name":"Contijoch M","last_name":null,"full_name":null},{"first_name":"Cuberes R","last_name":null,"full_name":null},{"first_name":"D\u00edaz JL","last_name":null,"full_name":null},{"first_name":"Fern\u00e1ndez A","last_name":null,"full_name":null},{"first_name":"Holenz J","last_name":null,"full_name":null},{"first_name":"Laggner C","last_name":null,"full_name":null},{"first_name":"Merlos M","last_name":null,"full_name":null},{"first_name":"Port A","last_name":null,"full_name":null},{"first_name":"Serafini MT","last_name":null,"full_name":null},{"first_name":"Vela JM","last_name":null,"full_name":null},{"first_name":"Zamanillo D","last_name":null,"full_name":null},{"first_name":"Almansa C.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3870","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3870","created_at":"2024-05-21T20:13:49.000000Z","updated_at":null}}