{"data":{"id":3713,"citation":"Lampe JW, Alford JS, Boriak-Sjodin PA, Brach D, Cosmopoulos K, Duncan KW, Eckley ST, Foley MA, Harvey DM, Motwani V, Munchhof MJ, Raimondi A, Riera TV, Tang C, Thomenius MJ, Totman J, Farrow NA.: Discovery of a First-in-Class Inhibitor of the Histone Methyltransferase SETD2 Suitable for Preclinical Studies. ACS Med Chem Lett, Volume 12 (10), 2021","title":"Discovery of a First-in-Class Inhibitor of the Histone Methyltransferase SETD2 Suitable for Preclinical Studies.","doi":"10.1021\/acsmedchemlett.1c00272","doi_url":"https:\/\/doi.org\/10.1021\/acsmedchemlett.1c00272","pmid":"34671445","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/34671445\/","year":2021,"journal":"ACS Med Chem Lett","volume":"12","issue":"10","page":"1539-1545","authors":[{"first_name":"Alford JS","last_name":null,"full_name":null},{"first_name":"Boriak-Sjodin PA","last_name":null,"full_name":null},{"first_name":"Brach D","last_name":null,"full_name":null},{"first_name":"Cosmopoulos K","last_name":null,"full_name":null},{"first_name":"Duncan KW","last_name":null,"full_name":null},{"first_name":"Eckley ST","last_name":null,"full_name":null},{"first_name":"Farrow NA.","last_name":null,"full_name":null},{"first_name":"Foley MA","last_name":null,"full_name":null},{"first_name":"Harvey DM","last_name":null,"full_name":null},{"first_name":"Lampe JW","last_name":null,"full_name":null},{"first_name":"Motwani V","last_name":null,"full_name":null},{"first_name":"Munchhof MJ","last_name":null,"full_name":null},{"first_name":"Raimondi A","last_name":null,"full_name":null},{"first_name":"Riera TV","last_name":null,"full_name":null},{"first_name":"Tang C","last_name":null,"full_name":null},{"first_name":"Thomenius MJ","last_name":null,"full_name":null},{"first_name":"Totman J","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3713","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3713","created_at":"2024-05-21T20:13:04.000000Z","updated_at":null}}