{"data":{"id":3684,"citation":"Andersson V, Bergstr\u00f6m F, Br\u00e5nalt J, Gr\u00f6nberg G, Gustafsson D, Karlsson S, Polla M, Bergman J, Kihlberg J.: Macrocyclic Prodrugs of a Selective Nonpeptidic Direct Thrombin Inhibitor Display High Permeability, Efficient Bioconversion but Low Bioavailability. J Med Chem, Volume 59 (14), 2016","title":"Macrocyclic Prodrugs of a Selective Nonpeptidic Direct Thrombin Inhibitor Display High Permeability, Efficient Bioconversion but Low Bioavailability.","doi":"10.1021\/acs.jmedchem.5b01871","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.5b01871","pmid":"27347787","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/27347787\/","year":2016,"journal":"J Med Chem","volume":"59","issue":"14","page":"6658-6670","authors":[{"first_name":"Andersson V","last_name":null,"full_name":null},{"first_name":"Bergman J","last_name":null,"full_name":null},{"first_name":"Bergstr\u00f6m F","last_name":null,"full_name":null},{"first_name":"Br\u00e5nalt J","last_name":null,"full_name":null},{"first_name":"Gr\u00f6nberg G","last_name":null,"full_name":null},{"first_name":"Gustafsson D","last_name":null,"full_name":null},{"first_name":"Karlsson S","last_name":null,"full_name":null},{"first_name":"Kihlberg J.","last_name":null,"full_name":null},{"first_name":"Polla M","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3684","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3684","created_at":"2024-05-21T20:12:56.000000Z","updated_at":null}}