{"data":{"id":3653,"citation":"Nakajima R, Oono H, Sugiyama S, Matsueda Y, Ida T, Kakuda S, Hirata J, Baba A, Makino A, Matsuyama R, White RD, Wurz R\u03a1, Shin Y, Min X, Guzman-Perez A, Wang Z, Symons A, Singh SK, Mothe SR, Belyakov S, Chakrabarti A, Shuto S.: Discovery of [1,2,4]Triazolo[1,5-<i>a<\/i>]pyridine Derivatives as Potent and Orally Bioavailable ROR\u03b3t Inverse Agonists. ACS Med Chem Lett, Volume 11 (4), 2020","title":"Discovery of [1,2,4]Triazolo[1,5-<i>a<\/i>]pyridine Derivatives as Potent and Orally Bioavailable ROR\u03b3t Inverse Agonists.","doi":"10.1021\/acsmedchemlett.9b00649","doi_url":"https:\/\/doi.org\/10.1021\/acsmedchemlett.9b00649","pmid":"32292560","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/32292560\/","year":2020,"journal":"ACS Med Chem Lett","volume":"11","issue":"4","page":"528-534","authors":[{"first_name":"Baba A","last_name":null,"full_name":null},{"first_name":"Belyakov S","last_name":null,"full_name":null},{"first_name":"Chakrabarti A","last_name":null,"full_name":null},{"first_name":"Guzman-Perez A","last_name":null,"full_name":null},{"first_name":"Hirata J","last_name":null,"full_name":null},{"first_name":"Ida T","last_name":null,"full_name":null},{"first_name":"Kakuda S","last_name":null,"full_name":null},{"first_name":"Makino A","last_name":null,"full_name":null},{"first_name":"Matsueda Y","last_name":null,"full_name":null},{"first_name":"Matsuyama R","last_name":null,"full_name":null},{"first_name":"Min X","last_name":null,"full_name":null},{"first_name":"Mothe SR","last_name":null,"full_name":null},{"first_name":"Nakajima R","last_name":null,"full_name":null},{"first_name":"Oono H","last_name":null,"full_name":null},{"first_name":"Shin Y","last_name":null,"full_name":null},{"first_name":"Shuto S.","last_name":null,"full_name":null},{"first_name":"Singh SK","last_name":null,"full_name":null},{"first_name":"Sugiyama S","last_name":null,"full_name":null},{"first_name":"Symons A","last_name":null,"full_name":null},{"first_name":"Wang Z","last_name":null,"full_name":null},{"first_name":"White RD","last_name":null,"full_name":null},{"first_name":"Wurz R\u03a1","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3653","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3653","created_at":"2024-05-21T20:12:50.000000Z","updated_at":null}}