{"data":{"id":3552,"citation":"Yang MG, Beaudoin-Bertrand M, Xiao Z, Marcoux D, Weigelt CA, Yip S, Wu DR, Ruzanov M, Sack JS, Wang J, Yarde M, Li S, Shuster DJ, Xie JH, Sherry T, Obermeier MT, Fura A, Stefanski K, Cornelius G, Khandelwal P, Karmakar A, Basha M, Babu V, Gupta AK, Mathur A, Salter-Cid L, Denton R, Zhao Q, Dhar TGM.: Tricyclic-Carbocyclic ROR\u03b3t Inverse Agonists-Discovery of BMS-986313. J Med Chem, Volume 64 (5), 2021","title":"Tricyclic-Carbocyclic ROR\u03b3t Inverse Agonists-Discovery of BMS-986313.","doi":"10.1021\/acs.jmedchem.0c01992","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.0c01992","pmid":"33591748","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/33591748\/","year":2021,"journal":"J Med Chem","volume":"64","issue":"5","page":"2714-2724","authors":[{"first_name":"Babu V","last_name":null,"full_name":null},{"first_name":"Basha M","last_name":null,"full_name":null},{"first_name":"Beaudoin-Bertrand M","last_name":null,"full_name":null},{"first_name":"Cornelius G","last_name":null,"full_name":null},{"first_name":"Denton R","last_name":null,"full_name":null},{"first_name":"Dhar TGM.","last_name":null,"full_name":null},{"first_name":"Fura A","last_name":null,"full_name":null},{"first_name":"Gupta AK","last_name":null,"full_name":null},{"first_name":"Karmakar A","last_name":null,"full_name":null},{"first_name":"Khandelwal P","last_name":null,"full_name":null},{"first_name":"Li S","last_name":null,"full_name":null},{"first_name":"Marcoux D","last_name":null,"full_name":null},{"first_name":"Mathur A","last_name":null,"full_name":null},{"first_name":"Obermeier MT","last_name":null,"full_name":null},{"first_name":"Ruzanov M","last_name":null,"full_name":null},{"first_name":"Sack JS","last_name":null,"full_name":null},{"first_name":"Salter-Cid L","last_name":null,"full_name":null},{"first_name":"Sherry T","last_name":null,"full_name":null},{"first_name":"Shuster DJ","last_name":null,"full_name":null},{"first_name":"Stefanski K","last_name":null,"full_name":null},{"first_name":"Wang J","last_name":null,"full_name":null},{"first_name":"Weigelt CA","last_name":null,"full_name":null},{"first_name":"Wu DR","last_name":null,"full_name":null},{"first_name":"Xiao Z","last_name":null,"full_name":null},{"first_name":"Xie JH","last_name":null,"full_name":null},{"first_name":"Yang MG","last_name":null,"full_name":null},{"first_name":"Yarde M","last_name":null,"full_name":null},{"first_name":"Yip S","last_name":null,"full_name":null},{"first_name":"Zhao Q","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3552","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3552","created_at":"2024-05-21T20:12:28.000000Z","updated_at":null}}