{"data":{"id":3533,"citation":"Cherney RJ, Cornelius LAM, Srivastava A, Weigelt CA, Marcoux D, Duan JJ, Shi Q, Batt DG, Liu Q, Yip S, Wu DR, Ruzanov M, Sack J, Khan J, Wang J, Yarde M, Cvijic ME, Mathur A, Li S, Shuster D, Khandelwal P, Borowski V, Xie J, Obermeier M, Fura A, Stefanski K, Cornelius G, Tino JA, Macor JE, Salter-Cid L, Denton R, Zhao Q, Carter PH, Dhar TGM.: Discovery of BMS-986251: A Clinically Viable, Potent, and Selective ROR\u03b3t Inverse Agonist. ACS Med Chem Lett, Volume 11 (6), 2020","title":"Discovery of BMS-986251: A Clinically Viable, Potent, and Selective ROR\u03b3t Inverse Agonist.","doi":"10.1021\/acsmedchemlett.0c00063","doi_url":"https:\/\/doi.org\/10.1021\/acsmedchemlett.0c00063","pmid":"32551004","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/32551004\/","year":2020,"journal":"ACS Med Chem Lett","volume":"11","issue":"6","page":"1221-1227","authors":[{"first_name":"Batt DG","last_name":null,"full_name":null},{"first_name":"Borowski V","last_name":null,"full_name":null},{"first_name":"Carter PH","last_name":null,"full_name":null},{"first_name":"Cherney RJ","last_name":null,"full_name":null},{"first_name":"Cornelius G","last_name":null,"full_name":null},{"first_name":"Cornelius LAM","last_name":null,"full_name":null},{"first_name":"Cvijic ME","last_name":null,"full_name":null},{"first_name":"Denton R","last_name":null,"full_name":null},{"first_name":"Dhar TGM.","last_name":null,"full_name":null},{"first_name":"Duan JJ","last_name":null,"full_name":null},{"first_name":"Fura A","last_name":null,"full_name":null},{"first_name":"Khan J","last_name":null,"full_name":null},{"first_name":"Khandelwal P","last_name":null,"full_name":null},{"first_name":"Li S","last_name":null,"full_name":null},{"first_name":"Liu Q","last_name":null,"full_name":null},{"first_name":"Macor JE","last_name":null,"full_name":null},{"first_name":"Marcoux D","last_name":null,"full_name":null},{"first_name":"Mathur A","last_name":null,"full_name":null},{"first_name":"Obermeier M","last_name":null,"full_name":null},{"first_name":"Ruzanov M","last_name":null,"full_name":null},{"first_name":"Sack J","last_name":null,"full_name":null},{"first_name":"Salter-Cid L","last_name":null,"full_name":null},{"first_name":"Shi Q","last_name":null,"full_name":null},{"first_name":"Shuster D","last_name":null,"full_name":null},{"first_name":"Srivastava A","last_name":null,"full_name":null},{"first_name":"Stefanski K","last_name":null,"full_name":null},{"first_name":"Tino JA","last_name":null,"full_name":null},{"first_name":"Wang J","last_name":null,"full_name":null},{"first_name":"Weigelt CA","last_name":null,"full_name":null},{"first_name":"Wu DR","last_name":null,"full_name":null},{"first_name":"Xie J","last_name":null,"full_name":null},{"first_name":"Yarde M","last_name":null,"full_name":null},{"first_name":"Yip S","last_name":null,"full_name":null},{"first_name":"Zhao Q","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3533","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3533","created_at":"2024-05-21T20:12:24.000000Z","updated_at":null}}