{"data":{"id":3472,"citation":"Munck Af Rosensch\u00f6ld M, Johannesson P, Nikitidis A, Tyrchan C, Chang HF, R\u00f6nn R, Chapman D, Ullah V, Nikitidis G, Glader P, K\u00e4ck H, Bonn B, W\u00e5gberg F, Bj\u00f6rkstrand E, Andersson U, Swedin L, Rohman M, Andreasson T, Bergstr\u00f6m EL, Jiang F, Zhou XH, Lundqvist AJ, Malmberg A, Ek M, Gordon E, Pettersen A, Ripa L, Davis AM.: Discovery of the Oral Leukotriene C4 Synthase Inhibitor (1<i>S<\/i>,2<i>S<\/i>)-2-({5-[(5-Chloro-2,4-difluorophenyl)(2-fluoro-2-methylpropyl)amino]-3-methoxypyrazin-2-yl}carbonyl)cyclopropanecarboxylic Acid (AZD9898) as a New Treatment for Asthma. J Med Chem, Volume 62 (17), 2019","title":"Discovery of the Oral Leukotriene C4 Synthase Inhibitor (1<i>S<\/i>,2<i>S<\/i>)-2-({5-[(5-Chloro-2,4-difluorophenyl)(2-fluoro-2-methylpropyl)amino]-3-methoxypyrazin-2-yl}carbonyl)cyclopropanecarboxylic Acid (AZD9898) as a New Treatment for Asthma.","doi":"10.1021\/acs.jmedchem.9b00555","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.9b00555","pmid":"31415176","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/31415176\/","year":2019,"journal":"J Med Chem","volume":"62","issue":"17","page":"7769-7787","authors":[{"first_name":"Andersson U","last_name":null,"full_name":null},{"first_name":"Andreasson T","last_name":null,"full_name":null},{"first_name":"Bergstr\u00f6m EL","last_name":null,"full_name":null},{"first_name":"Bj\u00f6rkstrand E","last_name":null,"full_name":null},{"first_name":"Bonn B","last_name":null,"full_name":null},{"first_name":"Chang HF","last_name":null,"full_name":null},{"first_name":"Chapman D","last_name":null,"full_name":null},{"first_name":"Davis AM.","last_name":null,"full_name":null},{"first_name":"Ek M","last_name":null,"full_name":null},{"first_name":"Glader P","last_name":null,"full_name":null},{"first_name":"Gordon E","last_name":null,"full_name":null},{"first_name":"Jiang F","last_name":null,"full_name":null},{"first_name":"Johannesson P","last_name":null,"full_name":null},{"first_name":"K\u00e4ck H","last_name":null,"full_name":null},{"first_name":"Lundqvist AJ","last_name":null,"full_name":null},{"first_name":"Malmberg A","last_name":null,"full_name":null},{"first_name":"Munck Af Rosensch\u00f6ld M","last_name":null,"full_name":null},{"first_name":"Nikitidis A","last_name":null,"full_name":null},{"first_name":"Nikitidis G","last_name":null,"full_name":null},{"first_name":"Pettersen A","last_name":null,"full_name":null},{"first_name":"Ripa L","last_name":null,"full_name":null},{"first_name":"Rohman M","last_name":null,"full_name":null},{"first_name":"R\u00f6nn R","last_name":null,"full_name":null},{"first_name":"Swedin L","last_name":null,"full_name":null},{"first_name":"Tyrchan C","last_name":null,"full_name":null},{"first_name":"Ullah V","last_name":null,"full_name":null},{"first_name":"W\u00e5gberg F","last_name":null,"full_name":null},{"first_name":"Zhou XH","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3472","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3472","created_at":"2024-05-21T20:12:12.000000Z","updated_at":null}}