{"data":{"id":3439,"citation":"Palmer WS, Poncet-Montange G, Liu G, Petrocchi A, Reyna N, Subramanian G, Theroff J, Yau A, Kost-Alimova M, Bardenhagen JP, Leo E, Shepard HE, Tieu TN, Shi X, Zhan Y, Zhao S, Barton MC, Draetta G, Toniatti C, Jones P, Geck Do M, Andersen JN.: Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor. J Med Chem, Volume 59 (4), 2016","title":"Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor.","doi":"10.1021\/acs.jmedchem.5b00405","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.5b00405","pmid":"26061247","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/26061247\/","year":2016,"journal":"J Med Chem","volume":"59","issue":"4","page":"1440-1454","authors":[{"first_name":"Andersen JN.","last_name":null,"full_name":null},{"first_name":"Bardenhagen JP","last_name":null,"full_name":null},{"first_name":"Barton MC","last_name":null,"full_name":null},{"first_name":"Draetta G","last_name":null,"full_name":null},{"first_name":"Geck Do M","last_name":null,"full_name":null},{"first_name":"Jones P","last_name":null,"full_name":null},{"first_name":"Kost-Alimova M","last_name":null,"full_name":null},{"first_name":"Leo E","last_name":null,"full_name":null},{"first_name":"Liu G","last_name":null,"full_name":null},{"first_name":"Palmer WS","last_name":null,"full_name":null},{"first_name":"Petrocchi A","last_name":null,"full_name":null},{"first_name":"Poncet-Montange G","last_name":null,"full_name":null},{"first_name":"Reyna N","last_name":null,"full_name":null},{"first_name":"Shepard HE","last_name":null,"full_name":null},{"first_name":"Shi X","last_name":null,"full_name":null},{"first_name":"Subramanian G","last_name":null,"full_name":null},{"first_name":"Theroff J","last_name":null,"full_name":null},{"first_name":"Tieu TN","last_name":null,"full_name":null},{"first_name":"Toniatti C","last_name":null,"full_name":null},{"first_name":"Yau A","last_name":null,"full_name":null},{"first_name":"Zhan Y","last_name":null,"full_name":null},{"first_name":"Zhao S","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3439","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3439","created_at":"2024-05-21T20:12:05.000000Z","updated_at":null}}