{"data":{"id":3401,"citation":"Garc\u00eda M, Virgili M, Alonso M, Alegret C, Farran J, Fern\u00e1ndez B, Bordas M, Pascual R, Burgue\u00f1o J, Vidal-Torres A, Fern\u00e1ndez de Henestrosa AR, Ayet E, Merlos M, Vela JM, Plata-Salam\u00e1n CR, Almansa C.: Discovery of EST73502, a Dual \u03bc-Opioid Receptor Agonist and \u03c3<sub>1<\/sub> Receptor Antagonist Clinical Candidate for the Treatment of Pain. J Med Chem, Volume 63 (24), 2020","title":"Discovery of EST73502, a Dual \u03bc-Opioid Receptor Agonist and \u03c3<sub>1<\/sub> Receptor Antagonist Clinical Candidate for the Treatment of Pain.","doi":"10.1021\/acs.jmedchem.0c01127","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.0c01127","pmid":"33064947","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/33064947\/","year":2020,"journal":"J Med Chem","volume":"63","issue":"24","page":"15508-15526","authors":[{"first_name":"Alegret C","last_name":null,"full_name":null},{"first_name":"Almansa C.","last_name":null,"full_name":null},{"first_name":"Alonso M","last_name":null,"full_name":null},{"first_name":"Ayet E","last_name":null,"full_name":null},{"first_name":"Bordas M","last_name":null,"full_name":null},{"first_name":"Burgue\u00f1o J","last_name":null,"full_name":null},{"first_name":"Farran J","last_name":null,"full_name":null},{"first_name":"Fern\u00e1ndez B","last_name":null,"full_name":null},{"first_name":"Fern\u00e1ndez de Henestrosa AR","last_name":null,"full_name":null},{"first_name":"Garcia M","last_name":null,"full_name":null},{"first_name":"Merlos M","last_name":null,"full_name":null},{"first_name":"Pascual R","last_name":null,"full_name":null},{"first_name":"Plata-Salam\u00e1n CR","last_name":null,"full_name":null},{"first_name":"Vela JM","last_name":null,"full_name":null},{"first_name":"Vidal-Torres A","last_name":null,"full_name":null},{"first_name":"Virgili M","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3401","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3401","created_at":"2024-05-21T20:11:57.000000Z","updated_at":null}}