{"data":{"id":3399,"citation":"Quancard J, Simic O, Pissot Soldermann C, Aichholz R, Blatter M, Renatus M, Erbel P, Melkko S, Endres R, Sorge M, Kieffer L, Wagner T, Beltz K, Mcsheehy P, Wartmann M, R\u00e9gnier CH, Calzascia T, Radimerski T, Bigaud M, Weiss A, Bornancin F, Schlapbach A.: Optimization of the <i>In Vivo<\/i> Potency of Pyrazolopyrimidine MALT1 Protease Inhibitors by Reducing Metabolism and Increasing Potency in Whole Blood. J Med Chem, Volume 63 (23), 2020","title":"Optimization of the <i>In Vivo<\/i> Potency of Pyrazolopyrimidine MALT1 Protease Inhibitors by Reducing Metabolism and Increasing Potency in Whole Blood.","doi":"10.1021\/acs.jmedchem.0c01246","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.0c01246","pmid":"33216547","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/33216547\/","year":2020,"journal":"J Med Chem","volume":"63","issue":"23","page":"14594-14608","authors":[{"first_name":"Aichholz R","last_name":null,"full_name":null},{"first_name":"Beltz K","last_name":null,"full_name":null},{"first_name":"Bigaud M","last_name":null,"full_name":null},{"first_name":"Blatter M","last_name":null,"full_name":null},{"first_name":"Bornancin F","last_name":null,"full_name":null},{"first_name":"Calzascia T","last_name":null,"full_name":null},{"first_name":"Endres R","last_name":null,"full_name":null},{"first_name":"Erbel P","last_name":null,"full_name":null},{"first_name":"Kieffer L","last_name":null,"full_name":null},{"first_name":"Mcsheehy P","last_name":null,"full_name":null},{"first_name":"Melkko S","last_name":null,"full_name":null},{"first_name":"Pissot Soldermann C","last_name":null,"full_name":null},{"first_name":"Quancard J","last_name":null,"full_name":null},{"first_name":"Radimerski T","last_name":null,"full_name":null},{"first_name":"R\u00e9gnier CH","last_name":null,"full_name":null},{"first_name":"Renatus M","last_name":null,"full_name":null},{"first_name":"Schlapbach A.","last_name":null,"full_name":null},{"first_name":"Simic O","last_name":null,"full_name":null},{"first_name":"Sorge M","last_name":null,"full_name":null},{"first_name":"Wagner T","last_name":null,"full_name":null},{"first_name":"Wartmann M","last_name":null,"full_name":null},{"first_name":"Weiss A","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3399","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3399","created_at":"2024-05-21T20:11:57.000000Z","updated_at":null}}