{"data":{"id":3396,"citation":"Harcken C, Csengery J, Turner M, Wu L, Liang S, Sibley R, Brunette S, Labadia M, Hoyt K, Wayne A, Wieckowski T, Davis G, Panzenbeck M, Souza D, Kugler S, Terenzio D, Collin D, Smith D, Fryer RM, Tseng YC, Hehn JP, Fletcher K, Hughes RO.: Discovery of a Series of Pyrazinone ROR\u03b3 Antagonists and Identification of the Clinical Candidate BI 730357. ACS Med Chem Lett, Volume 12 (1), 2021","title":"Discovery of a Series of Pyrazinone ROR\u03b3 Antagonists and Identification of the Clinical Candidate BI 730357.","doi":"10.1021\/acsmedchemlett.0c00575","doi_url":"https:\/\/doi.org\/10.1021\/acsmedchemlett.0c00575","pmid":"33488976","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/33488976\/","year":2021,"journal":"ACS Med Chem Lett","volume":"12","issue":"1","page":"143-154","authors":[{"first_name":"Brunette S","last_name":null,"full_name":null},{"first_name":"Collin D","last_name":null,"full_name":null},{"first_name":"Csengery J","last_name":null,"full_name":null},{"first_name":"Davis G","last_name":null,"full_name":null},{"first_name":"Fletcher K","last_name":null,"full_name":null},{"first_name":"Fryer RM","last_name":null,"full_name":null},{"first_name":"Harcken C","last_name":null,"full_name":null},{"first_name":"Hehn JP","last_name":null,"full_name":null},{"first_name":"Hoyt K","last_name":null,"full_name":null},{"first_name":"Hughes RO.","last_name":null,"full_name":null},{"first_name":"Kugler S","last_name":null,"full_name":null},{"first_name":"Labadia M","last_name":null,"full_name":null},{"first_name":"Liang S","last_name":null,"full_name":null},{"first_name":"Panzenbeck M","last_name":null,"full_name":null},{"first_name":"Sibley R","last_name":null,"full_name":null},{"first_name":"Smith D","last_name":null,"full_name":null},{"first_name":"Souza D","last_name":null,"full_name":null},{"first_name":"Terenzio D","last_name":null,"full_name":null},{"first_name":"Tseng YC","last_name":null,"full_name":null},{"first_name":"Turner M","last_name":null,"full_name":null},{"first_name":"Wayne A","last_name":null,"full_name":null},{"first_name":"Wieckowski T","last_name":null,"full_name":null},{"first_name":"Wu L","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3396","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3396","created_at":"2024-05-21T20:11:56.000000Z","updated_at":null}}