{"data":{"id":3388,"citation":"Duan JJ, Lu Z, Jiang B, Stachura S, Weigelt CA, Sack JS, Khan J, Ruzanov M, Galella MA, Wu DR, Yarde M, Shen DR, Shuster DJ, Borowski V, Xie JH, Zhang L, Vanteru S, Gupta AK, Mathur A, Zhao Q, Foster W, Salter-Cid LM, Carter PH, Dhar TGM.: Structure-based Discovery of Phenyl (3-Phenylpyrrolidin-3-yl)sulfones as Selective, Orally Active ROR\u03b3t Inverse Agonists. ACS Med Chem Lett, Volume 10 (3), 2019","title":"Structure-based Discovery of Phenyl (3-Phenylpyrrolidin-3-yl)sulfones as Selective, Orally Active ROR\u03b3t Inverse Agonists.","doi":"10.1021\/acsmedchemlett.9b00010","doi_url":"https:\/\/doi.org\/10.1021\/acsmedchemlett.9b00010","pmid":"30891142","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/30891142\/","year":2019,"journal":"ACS Med Chem Lett","volume":"10","issue":"3","page":"367-373","authors":[{"first_name":"Borowski V","last_name":null,"full_name":null},{"first_name":"Carter PH","last_name":null,"full_name":null},{"first_name":"Dhar TGM.","last_name":null,"full_name":null},{"first_name":"Duan JJ","last_name":null,"full_name":null},{"first_name":"Foster W","last_name":null,"full_name":null},{"first_name":"Galella MA","last_name":null,"full_name":null},{"first_name":"Gupta AK","last_name":null,"full_name":null},{"first_name":"Jiang B","last_name":null,"full_name":null},{"first_name":"Khan J","last_name":null,"full_name":null},{"first_name":"Lu Z","last_name":null,"full_name":null},{"first_name":"Mathur A","last_name":null,"full_name":null},{"first_name":"Ruzanov M","last_name":null,"full_name":null},{"first_name":"Sack JS","last_name":null,"full_name":null},{"first_name":"Salter-Cid LM","last_name":null,"full_name":null},{"first_name":"Shen DR","last_name":null,"full_name":null},{"first_name":"Shuster DJ","last_name":null,"full_name":null},{"first_name":"Stachura S","last_name":null,"full_name":null},{"first_name":"Vanteru S","last_name":null,"full_name":null},{"first_name":"Weigelt CA","last_name":null,"full_name":null},{"first_name":"Wu DR","last_name":null,"full_name":null},{"first_name":"Xie JH","last_name":null,"full_name":null},{"first_name":"Yarde M","last_name":null,"full_name":null},{"first_name":"Zhang L","last_name":null,"full_name":null},{"first_name":"Zhao Q","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3388","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3388","created_at":"2024-05-21T20:11:55.000000Z","updated_at":null}}