{"data":{"id":3364,"citation":"Rankovic Z, Cai J, Kerr J, Fradera X, Robinson J, Mistry A, Finlay W, McGarry G, Andrews F, Caulfield W, Cumming I, Dempster M, Waller J, Arbuckle W, Anderson M, Martin I, Mitchell A, Long C, Baugh M, Westwood P, Kinghorn E, Jones P, Uitdehaag JC, van Zeeland M, Potin D, Saniere L, Fouquet A, Chevallier F, Deronzier H, Dorleans C, Nicolai E.: Optimisation of 2-cyano-pyrimidine inhibitors of cathepsin K: improving selectivity over hERG. Bioorg Med Chem Lett, Volume 20 (21), 2010","title":"Optimisation of 2-cyano-pyrimidine inhibitors of cathepsin K: improving selectivity over hERG.","doi":"10.1016\/j.bmcl.2010.08.101","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2010.08.101","pmid":"20843687","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20843687\/","year":2010,"journal":"Bioorg Med Chem Lett","volume":"20","issue":"21","page":"6237-6241","authors":[{"first_name":"Anderson M","last_name":null,"full_name":null},{"first_name":"Andrews F","last_name":null,"full_name":null},{"first_name":"Arbuckle W","last_name":null,"full_name":null},{"first_name":"Baugh M","last_name":null,"full_name":null},{"first_name":"Cai J","last_name":null,"full_name":null},{"first_name":"Caulfield W","last_name":null,"full_name":null},{"first_name":"Chevallier F","last_name":null,"full_name":null},{"first_name":"Cumming I","last_name":null,"full_name":null},{"first_name":"Dempster M","last_name":null,"full_name":null},{"first_name":"Deronzier H","last_name":null,"full_name":null},{"first_name":"Dorleans C","last_name":null,"full_name":null},{"first_name":"Finlay W","last_name":null,"full_name":null},{"first_name":"Fouquet A","last_name":null,"full_name":null},{"first_name":"Fradera X","last_name":null,"full_name":null},{"first_name":"Jones P","last_name":null,"full_name":null},{"first_name":"Kerr J","last_name":null,"full_name":null},{"first_name":"Kinghorn E","last_name":null,"full_name":null},{"first_name":"Long C","last_name":null,"full_name":null},{"first_name":"Martin I","last_name":null,"full_name":null},{"first_name":"McGarry G","last_name":null,"full_name":null},{"first_name":"Mistry A","last_name":null,"full_name":null},{"first_name":"Mitchell A","last_name":null,"full_name":null},{"first_name":"Nicolai E.","last_name":null,"full_name":null},{"first_name":"Potin D","last_name":null,"full_name":null},{"first_name":"Rankovic Z","last_name":null,"full_name":null},{"first_name":"Robinson J","last_name":null,"full_name":null},{"first_name":"Saniere L","last_name":null,"full_name":null},{"first_name":"Uitdehaag JC","last_name":null,"full_name":null},{"first_name":"van Zeeland M","last_name":null,"full_name":null},{"first_name":"Waller J","last_name":null,"full_name":null},{"first_name":"Westwood P","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3364","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3364","created_at":"2024-05-21T20:11:50.000000Z","updated_at":null}}