{"data":{"id":3363,"citation":"Eggert E, Hillig RC, Koehr S, St\u00f6ckigt D, Weiske J, Barak N, Mowat J, Brumby T, Christ CD, Ter Laak A, Lang T, Fernandez-Montalvan AE, Badock V, Weinmann H, Hartung IV, Barsyte-Lovejoy D, Szewczyk M, Kennedy S, Li F, Vedadi M, Brown PJ, Santhakumar V, Arrowsmith CH, Stellfeld T, Stresemann C.: Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2. J Med Chem, Volume 59 (10), 2016","title":"Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2.","doi":"10.1021\/acs.jmedchem.5b01890","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.5b01890","pmid":"27075367","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/27075367\/","year":2016,"journal":"J Med Chem","volume":"59","issue":"10","page":"4578-4600","authors":[{"first_name":"Arrowsmith CH","last_name":null,"full_name":null},{"first_name":"Badock V","last_name":null,"full_name":null},{"first_name":"Barak N","last_name":null,"full_name":null},{"first_name":"Barsyte-Lovejoy D","last_name":null,"full_name":null},{"first_name":"Brown PJ","last_name":null,"full_name":null},{"first_name":"Brumby T","last_name":null,"full_name":null},{"first_name":"Christ CD","last_name":null,"full_name":null},{"first_name":"Eggert E","last_name":null,"full_name":null},{"first_name":"Fernandez-Montalvan AE","last_name":null,"full_name":null},{"first_name":"Hartung IV","last_name":null,"full_name":null},{"first_name":"Hillig RC","last_name":null,"full_name":null},{"first_name":"Kennedy S","last_name":null,"full_name":null},{"first_name":"Koehr S","last_name":null,"full_name":null},{"first_name":"Lang T","last_name":null,"full_name":null},{"first_name":"Li F","last_name":null,"full_name":null},{"first_name":"Mowat J","last_name":null,"full_name":null},{"first_name":"Santhakumar V","last_name":null,"full_name":null},{"first_name":"Stellfeld T","last_name":null,"full_name":null},{"first_name":"St\u00f6ckigt D","last_name":null,"full_name":null},{"first_name":"Stresemann C.","last_name":null,"full_name":null},{"first_name":"Szewczyk M","last_name":null,"full_name":null},{"first_name":"Ter Laak A","last_name":null,"full_name":null},{"first_name":"Vedadi M","last_name":null,"full_name":null},{"first_name":"Weinmann H","last_name":null,"full_name":null},{"first_name":"Weiske J","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3363","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3363","created_at":"2024-05-21T20:11:50.000000Z","updated_at":null}}