{"data":{"id":3348,"citation":"Sun ZY, Asberom T, Bara T, Bennett C, Burnett D, Chu I, Clader J, Cohen-Williams M, Cole D, Czarniecki M, Durkin J, Gallo G, Greenlee W, Josien H, Huang X, Hyde L, Jones N, Kazakevich I, Li H, Liu X, Lee J, Maccoss M, Mandal MB, McCracken T, Nomeir A, Mazzola R, Palani A, Parker EM, Pissarnitski DA, Qin J, Song L, Terracina G, Vicarel M, Voigt J, Xu R, Zhang L, Zhang Q, Zhao Z, Zhu X, Zhu Z.: Cyclic hydroxyamidines as amide isosteres: discovery of oxadiazolines and oxadiazines as potent and highly efficacious \u03b3-secretase modulators in vivo. J Med Chem, Volume 55 (1), 2012","title":"Cyclic hydroxyamidines as amide isosteres: discovery of oxadiazolines and oxadiazines as potent and highly efficacious \u03b3-secretase modulators in vivo.","doi":"10.1021\/jm201407j","doi_url":"https:\/\/doi.org\/10.1021\/jm201407j","pmid":"22098494","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/22098494\/","year":2012,"journal":"J Med Chem","volume":"55","issue":"1","page":"489-502","authors":[{"first_name":"Asberom T","last_name":null,"full_name":null},{"first_name":"Bara T","last_name":null,"full_name":null},{"first_name":"Bennett C","last_name":null,"full_name":null},{"first_name":"Burnett D","last_name":null,"full_name":null},{"first_name":"Chu I","last_name":null,"full_name":null},{"first_name":"Clader J","last_name":null,"full_name":null},{"first_name":"Cohen-Williams M","last_name":null,"full_name":null},{"first_name":"Cole D","last_name":null,"full_name":null},{"first_name":"Czarniecki M","last_name":null,"full_name":null},{"first_name":"Durkin J","last_name":null,"full_name":null},{"first_name":"Gallo G","last_name":null,"full_name":null},{"first_name":"Greenlee W","last_name":null,"full_name":null},{"first_name":"Huang X","last_name":null,"full_name":null},{"first_name":"Hyde L","last_name":null,"full_name":null},{"first_name":"Jones N","last_name":null,"full_name":null},{"first_name":"Josien H","last_name":null,"full_name":null},{"first_name":"Kazakevich I","last_name":null,"full_name":null},{"first_name":"Lee J","last_name":null,"full_name":null},{"first_name":"Li H","last_name":null,"full_name":null},{"first_name":"Liu X","last_name":null,"full_name":null},{"first_name":"Maccoss M","last_name":null,"full_name":null},{"first_name":"Mandal MB","last_name":null,"full_name":null},{"first_name":"Mazzola R","last_name":null,"full_name":null},{"first_name":"McCracken T","last_name":null,"full_name":null},{"first_name":"Nomeir A","last_name":null,"full_name":null},{"first_name":"Palani A","last_name":null,"full_name":null},{"first_name":"Parker EM","last_name":null,"full_name":null},{"first_name":"Pissarnitski DA","last_name":null,"full_name":null},{"first_name":"Qin J","last_name":null,"full_name":null},{"first_name":"Song L","last_name":null,"full_name":null},{"first_name":"Sun ZY","last_name":null,"full_name":null},{"first_name":"Terracina G","last_name":null,"full_name":null},{"first_name":"Vicarel M","last_name":null,"full_name":null},{"first_name":"Voigt J","last_name":null,"full_name":null},{"first_name":"Xu R","last_name":null,"full_name":null},{"first_name":"Zhang L","last_name":null,"full_name":null},{"first_name":"Zhang Q","last_name":null,"full_name":null},{"first_name":"Zhao Z","last_name":null,"full_name":null},{"first_name":"Zhu X","last_name":null,"full_name":null},{"first_name":"Zhu Z.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3348","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3348","created_at":"2024-05-21T20:11:47.000000Z","updated_at":null}}