{"data":{"id":3344,"citation":"Hoveyda HR, Marsault E, Gagnon R, Mathieu AP, V\u00e9zina M, Landry A, Wang Z, Benakli K, Beaubien S, Saint-Louis C, Brassard M, Pinault JF, Ouellet L, Bhat S, Ramaseshan M, Peng X, Foucher L, Beauchemin S, Bh\u00e9rer P, Veber DF, Peterson ML, Fraser GL.: Optimization of the potency and pharmacokinetic properties of a macrocyclic ghrelin receptor agonist (Part I): Development of ulimorelin (TZP-101) from hit to clinic. J Med Chem, Volume 54 (24), 2011","title":"Optimization of the potency and pharmacokinetic properties of a macrocyclic ghrelin receptor agonist (Part I): Development of ulimorelin (TZP-101) from hit to clinic.","doi":"10.1021\/jm2007062","doi_url":"https:\/\/doi.org\/10.1021\/jm2007062","pmid":"22106937","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/22106937\/","year":2011,"journal":"J Med Chem","volume":"54","issue":"24","page":"8305-8320","authors":[{"first_name":"Beaubien S","last_name":null,"full_name":null},{"first_name":"Beauchemin S","last_name":null,"full_name":null},{"first_name":"Benakli K","last_name":null,"full_name":null},{"first_name":"Bhat S","last_name":null,"full_name":null},{"first_name":"Bh\u00e9rer P","last_name":null,"full_name":null},{"first_name":"Brassard M","last_name":null,"full_name":null},{"first_name":"Foucher L","last_name":null,"full_name":null},{"first_name":"Fraser GL.","last_name":null,"full_name":null},{"first_name":"Gagnon R","last_name":null,"full_name":null},{"first_name":"Hoveyda HR","last_name":null,"full_name":null},{"first_name":"Landry A","last_name":null,"full_name":null},{"first_name":"Marsault E","last_name":null,"full_name":null},{"first_name":"Mathieu AP","last_name":null,"full_name":null},{"first_name":"Ouellet L","last_name":null,"full_name":null},{"first_name":"Peng X","last_name":null,"full_name":null},{"first_name":"Peterson ML","last_name":null,"full_name":null},{"first_name":"Pinault JF","last_name":null,"full_name":null},{"first_name":"Ramaseshan M","last_name":null,"full_name":null},{"first_name":"Saint-Louis C","last_name":null,"full_name":null},{"first_name":"Veber DF","last_name":null,"full_name":null},{"first_name":"V\u00e9zina M","last_name":null,"full_name":null},{"first_name":"Wang Z","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3344","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3344","created_at":"2024-05-21T20:11:46.000000Z","updated_at":null}}