{"data":{"id":3236,"citation":"Burch JD, Lau K, Barker JJ, Brookfield F, Chen Y, Chen Y, Eigenbrot C, Ellebrandt C, Ismaili MH, Johnson A, Kordt D, MacKinnon CH, McEwan PA, Ortwine DF, Stein DB, Wang X, Winkler D, Yuen PW, Zhang Y, Zarrin AA, Pei Z.: Property- and structure-guided discovery of a tetrahydroindazole series of interleukin-2 inducible T-cell kinase inhibitors. J Med Chem, Volume 57 (13), 2014","title":"Property- and structure-guided discovery of a tetrahydroindazole series of interleukin-2 inducible T-cell kinase inhibitors.","doi":"10.1021\/jm500550e","doi_url":"https:\/\/doi.org\/10.1021\/jm500550e","pmid":"24918870","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/24918870\/","year":2014,"journal":"J Med Chem","volume":"57","issue":"13","page":"5714-5727","authors":[{"first_name":"Barker JJ","last_name":null,"full_name":null},{"first_name":"Brookfield F","last_name":null,"full_name":null},{"first_name":"Burch JD","last_name":null,"full_name":null},{"first_name":"Chen Y","last_name":null,"full_name":null},{"first_name":"Eigenbrot C","last_name":null,"full_name":null},{"first_name":"Ellebrandt C","last_name":null,"full_name":null},{"first_name":"Ismaili MH","last_name":null,"full_name":null},{"first_name":"Johnson A","last_name":null,"full_name":null},{"first_name":"Kordt D","last_name":null,"full_name":null},{"first_name":"Lau K","last_name":null,"full_name":null},{"first_name":"MacKinnon CH","last_name":null,"full_name":null},{"first_name":"McEwan PA","last_name":null,"full_name":null},{"first_name":"Ortwine DF","last_name":null,"full_name":null},{"first_name":"Pei Z.","last_name":null,"full_name":null},{"first_name":"Stein DB","last_name":null,"full_name":null},{"first_name":"Wang X","last_name":null,"full_name":null},{"first_name":"Winkler D","last_name":null,"full_name":null},{"first_name":"Yuen PW","last_name":null,"full_name":null},{"first_name":"Zarrin AA","last_name":null,"full_name":null},{"first_name":"Zhang Y","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3236","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3236","created_at":"2024-05-21T09:16:29.000000Z","updated_at":null}}