{"data":{"id":3222,"citation":"Labadie S, Dragovich PS, Barrett K, Blair WS, Bergeron P, Chang C, Deshmukh G, Eigenbrot C, Ghilardi N, Gibbons P, Hurley CA, Johnson A, Kenny JR, Kohli PB, Kulagowski JJ, Liimatta M, Lupardus PJ, Mendonca R, Murray JM, Pulk R, Shia S, Steffek M, Ubhayakar S, Ultsch M, van Abbema A, Ward S, Zak M.: Structure-based discovery of C-2 substituted imidazo-pyrrolopyridine JAK1 inhibitors with improved selectivity over JAK2. Bioorg Med Chem Lett, Volume 22 (24), 2012","title":"Structure-based discovery of C-2 substituted imidazo-pyrrolopyridine JAK1 inhibitors with improved selectivity over JAK2.","doi":"10.1016\/j.bmcl.2012.10.008","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2012.10.008","pmid":"23107482","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/23107482\/","year":2012,"journal":"Bioorg Med Chem Lett","volume":"22","issue":"24","page":"7627-7633","authors":[{"first_name":"Barrett K","last_name":null,"full_name":null},{"first_name":"Bergeron P","last_name":null,"full_name":null},{"first_name":"Blair WS","last_name":null,"full_name":null},{"first_name":"Chang C","last_name":null,"full_name":null},{"first_name":"Deshmukh G","last_name":null,"full_name":null},{"first_name":"Dragovich PS","last_name":null,"full_name":null},{"first_name":"Eigenbrot C","last_name":null,"full_name":null},{"first_name":"Ghilardi N","last_name":null,"full_name":null},{"first_name":"Gibbons P","last_name":null,"full_name":null},{"first_name":"Hurley CA","last_name":null,"full_name":null},{"first_name":"Johnson A","last_name":null,"full_name":null},{"first_name":"Kenny JR","last_name":null,"full_name":null},{"first_name":"Kohli PB","last_name":null,"full_name":null},{"first_name":"Kulagowski JJ","last_name":null,"full_name":null},{"first_name":"Labadie S","last_name":null,"full_name":null},{"first_name":"Liimatta M","last_name":null,"full_name":null},{"first_name":"Lupardus PJ","last_name":null,"full_name":null},{"first_name":"Mendonca R","last_name":null,"full_name":null},{"first_name":"Murray JM","last_name":null,"full_name":null},{"first_name":"Pulk R","last_name":null,"full_name":null},{"first_name":"Shia S","last_name":null,"full_name":null},{"first_name":"Steffek M","last_name":null,"full_name":null},{"first_name":"Ubhayakar S","last_name":null,"full_name":null},{"first_name":"Ultsch M","last_name":null,"full_name":null},{"first_name":"van Abbema A","last_name":null,"full_name":null},{"first_name":"Ward S","last_name":null,"full_name":null},{"first_name":"Zak M.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3222","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3222","created_at":"2024-05-21T09:16:26.000000Z","updated_at":null}}