{"data":{"id":3058,"citation":"Ren\u00e9 O, Fauber BP, Barnard A, Chapman K, Deng Y, Eidenschenk C, Everett C, Gobbi A, Johnson AR, La H, Norman M, Salmon G, Summerhill S, Wong H.: Discovery of oxa-sultams as RORc inverse agonists showing reduced lipophilicity, improved selectivity and favorable ADME properties. Bioorg Med Chem Lett, Volume 26 (18), 2016","title":"Discovery of oxa-sultams as RORc inverse agonists showing reduced lipophilicity, improved selectivity and favorable ADME properties.","doi":"10.1016\/j.bmcl.2016.07.081","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2016.07.081","pmid":"27524313","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/27524313\/","year":2016,"journal":"Bioorg Med Chem Lett","volume":"26","issue":"18","page":"4455-4461","authors":[{"first_name":"Barnard A","last_name":null,"full_name":null},{"first_name":"Chapman K","last_name":null,"full_name":null},{"first_name":"Deng Y","last_name":null,"full_name":null},{"first_name":"Eidenschenk C","last_name":null,"full_name":null},{"first_name":"Everett C","last_name":null,"full_name":null},{"first_name":"Fauber BP","last_name":null,"full_name":null},{"first_name":"Gobbi A","last_name":null,"full_name":null},{"first_name":"Johnson AR","last_name":null,"full_name":null},{"first_name":"La H","last_name":null,"full_name":null},{"first_name":"Norman M","last_name":null,"full_name":null},{"first_name":"Ren\u00e9 O","last_name":null,"full_name":null},{"first_name":"Salmon G","last_name":null,"full_name":null},{"first_name":"Summerhill S","last_name":null,"full_name":null},{"first_name":"Wong H.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3058","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3058","created_at":"2024-05-21T09:15:45.000000Z","updated_at":null}}