{"data":{"id":3056,"citation":"Patel S, Harris SF, Gibbons P, Deshmukh G, Gustafson A, Kellar T, Lin H, Liu X, Liu Y, Liu Y, Ma C, Scearce-Levie K, Ghosh AS, Shin YG, Solanoy H, Wang J, Wang B, Yin J, Siu M, Lewcock JW.: Scaffold-Hopping and Structure-Based Discovery of Potent, Selective, And Brain Penetrant N-(1H-Pyrazol-3-yl)pyridin-2-amine Inhibitors of Dual Leucine Zipper Kinase (DLK, MAP3K12). J Med Chem, Volume 58 (20), 2015","title":"Scaffold-Hopping and Structure-Based Discovery of Potent, Selective, And Brain Penetrant N-(1H-Pyrazol-3-yl)pyridin-2-amine Inhibitors of Dual Leucine Zipper Kinase (DLK, MAP3K12).","doi":"10.1021\/acs.jmedchem.5b01072","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.5b01072","pmid":"26431428","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/26431428\/","year":2015,"journal":"J Med Chem","volume":"58","issue":"20","page":"8182-8199","authors":[{"first_name":"Deshmukh G","last_name":null,"full_name":null},{"first_name":"Ghosh AS","last_name":null,"full_name":null},{"first_name":"Gibbons P","last_name":null,"full_name":null},{"first_name":"Gustafson A","last_name":null,"full_name":null},{"first_name":"Harris SF","last_name":null,"full_name":null},{"first_name":"Kellar T","last_name":null,"full_name":null},{"first_name":"Lewcock JW.","last_name":null,"full_name":null},{"first_name":"Lin H","last_name":null,"full_name":null},{"first_name":"Liu X","last_name":null,"full_name":null},{"first_name":"Liu Y","last_name":null,"full_name":null},{"first_name":"Ma C","last_name":null,"full_name":null},{"first_name":"Patel S","last_name":null,"full_name":null},{"first_name":"Scearce-Levie K","last_name":null,"full_name":null},{"first_name":"Shin YG","last_name":null,"full_name":null},{"first_name":"Siu M","last_name":null,"full_name":null},{"first_name":"Solanoy H","last_name":null,"full_name":null},{"first_name":"Wang B","last_name":null,"full_name":null},{"first_name":"Wang J","last_name":null,"full_name":null},{"first_name":"Yin J","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3056","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3056","created_at":"2024-05-21T09:15:44.000000Z","updated_at":null}}