{"data":{"id":2940,"citation":"Kerns JK, Busch-Petersen J, Fu W, Boehm JC, Nie H, Muratore M, Bullion A, Lin G, Li H, Davis R, Lin X, Lakdawala AS, Cousins R, Field R, Payne J, Miller DD, Bamborough P, Christopher JA, Baldwin I, Osborn RR, Yonchuk J, Webb E, Rumsey WL.: 3,5-Disubstituted-indole-7-carboxamides as IKK\u03b2 Inhibitors: Optimization of Oral Activity via the C3 Substituent. ACS Med Chem Lett, Volume 9 (12), 2018","title":"3,5-Disubstituted-indole-7-carboxamides as IKK\u03b2 Inhibitors: Optimization of Oral Activity via the C3 Substituent.","doi":"10.1021\/acsmedchemlett.8b00291","doi_url":"https:\/\/doi.org\/10.1021\/acsmedchemlett.8b00291","pmid":"30613320","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/30613320\/","year":2018,"journal":"ACS Med Chem Lett","volume":"9","issue":"12","page":"1164-1169","authors":[{"first_name":"Baldwin I","last_name":null,"full_name":null},{"first_name":"Bamborough P","last_name":null,"full_name":null},{"first_name":"Boehm JC","last_name":null,"full_name":null},{"first_name":"Bullion A","last_name":null,"full_name":null},{"first_name":"Busch-Petersen J","last_name":null,"full_name":null},{"first_name":"Christopher JA","last_name":null,"full_name":null},{"first_name":"Cousins R","last_name":null,"full_name":null},{"first_name":"Davis R","last_name":null,"full_name":null},{"first_name":"Field R","last_name":null,"full_name":null},{"first_name":"Fu W","last_name":null,"full_name":null},{"first_name":"Kerns JK","last_name":null,"full_name":null},{"first_name":"Lakdawala AS","last_name":null,"full_name":null},{"first_name":"Li H","last_name":null,"full_name":null},{"first_name":"Lin G","last_name":null,"full_name":null},{"first_name":"Lin X","last_name":null,"full_name":null},{"first_name":"Miller DD","last_name":null,"full_name":null},{"first_name":"Muratore M","last_name":null,"full_name":null},{"first_name":"Nie H","last_name":null,"full_name":null},{"first_name":"Osborn RR","last_name":null,"full_name":null},{"first_name":"Payne J","last_name":null,"full_name":null},{"first_name":"Rumsey WL.","last_name":null,"full_name":null},{"first_name":"Webb E","last_name":null,"full_name":null},{"first_name":"Yonchuk J","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2940","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2940","created_at":"2023-06-23T15:10:18.000000Z","updated_at":null}}