{"data":{"id":282,"citation":"Asagarasu A, Matsui T, Hayashi H, Tamaoki S, Yamauchi Y, Minato K, Sato M.: Discovery of a novel 5-HT(3) antagonist\/5-HT(1A) agonist 3-amino-5,6,7,8-tetrahydro-2-{4-[4-(quinolin-2-yl)piperazin-1-yl]butyl}quinazolin-4(3H)-one (TZB-30878) as an orally bioavailable agent for irritable bowel syndrome. J Med Chem, Volume 53 (21), 2010","title":"Discovery of a novel 5-HT(3) antagonist\/5-HT(1A) agonist 3-amino-5,6,7,8-tetrahydro-2-{4-[4-(quinolin-2-yl)piperazin-1-yl]butyl}quinazolin-4(3H)-one (TZB-30878) as an orally bioavailable agent for irritable bowel syndrome.","doi":"10.1021\/jm1002292","doi_url":"https:\/\/doi.org\/10.1021\/jm1002292","pmid":"20931963","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20931963\/","year":2010,"journal":"J Med Chem","volume":"53","issue":"21","page":"7549-7563","authors":[{"first_name":"Asagarasu A","last_name":null,"full_name":null},{"first_name":"Hayashi H","last_name":null,"full_name":null},{"first_name":"Matsui T","last_name":null,"full_name":null},{"first_name":"Minato K","last_name":null,"full_name":null},{"first_name":"Sato M.","last_name":null,"full_name":null},{"first_name":"Tamaoki S","last_name":null,"full_name":null},{"first_name":"Yamauchi Y","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/282","landing_page":"https:\/\/molmedb.upol.cz\/publication\/282","created_at":"2020-06-29T09:51:21.000000Z","updated_at":null}}