{"data":{"id":2788,"citation":"Zanaletti R, Bettinetti L, Castaldo C, Cocconcelli G, Comery T, Dunlop J, Gaviraghi G, Ghiron C, Haydar SN, Jow F, Maccari L, Micco I, Nencini A, Scali C, Turlizzi E, Valacchi M.: Discovery of a novel alpha-7 nicotinic acetylcholine receptor agonist series and characterization of the potent, selective, and orally efficacious agonist 5-(4-acetyl[1,4]diazepan-1-yl)pentanoic acid [5-(4-methoxyphenyl)-1H-pyrazol-3-yl] amide (SEN15924, WAY-361789). J Med Chem, Volume 55 (10), 2012","title":"Discovery of a novel alpha-7 nicotinic acetylcholine receptor agonist series and characterization of the potent, selective, and orally efficacious agonist 5-(4-acetyl[1,4]diazepan-1-yl)pentanoic acid [5-(4-methoxyphenyl)-1H-pyrazol-3-yl] amide (SEN15924, WAY-361789).","doi":"10.1021\/jm300247y","doi_url":"https:\/\/doi.org\/10.1021\/jm300247y","pmid":"22468936","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/22468936\/","year":2012,"journal":"J Med Chem","volume":"55","issue":"10","page":"4806-4823","authors":[{"first_name":"Bettinetti L","last_name":null,"full_name":null},{"first_name":"Castaldo C","last_name":null,"full_name":null},{"first_name":"Cocconcelli G","last_name":null,"full_name":null},{"first_name":"Comery T","last_name":null,"full_name":null},{"first_name":"Dunlop J","last_name":null,"full_name":null},{"first_name":"Gaviraghi G","last_name":null,"full_name":null},{"first_name":"Ghiron C","last_name":null,"full_name":null},{"first_name":"Haydar SN","last_name":null,"full_name":null},{"first_name":"Jow F","last_name":null,"full_name":null},{"first_name":"Maccari L","last_name":null,"full_name":null},{"first_name":"Micco I","last_name":null,"full_name":null},{"first_name":"Nencini A","last_name":null,"full_name":null},{"first_name":"Scali C","last_name":null,"full_name":null},{"first_name":"Turlizzi E","last_name":null,"full_name":null},{"first_name":"Valacchi M.","last_name":null,"full_name":null},{"first_name":"Zanaletti R","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2788","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2788","created_at":"2023-06-23T15:09:44.000000Z","updated_at":null}}