{"data":{"id":2739,"citation":"Muthukaman N, Deshmukh S, Tambe M, Pisal D, Tondlekar S, Shaikh M, Sarode N, Kattige VG, Sawant P, Pisat M, Karande V, Honnegowda S, Kulkarni A, Behera D, Jadhav SB, Sangana RR, Gudi GS, Khairatkar-Joshi N, Gharat LA.: Alleviating CYP and hERG liabilities by structure optimization of dihydrofuran-fused tricyclic benzo[d]imidazole series - Potent, selective and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-2. Bioorg Med Chem Lett, Volume 28 (7), 2018","title":"Alleviating CYP and hERG liabilities by structure optimization of dihydrofuran-fused tricyclic benzo[d]imidazole series - Potent, selective and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-2.","doi":"10.1016\/j.bmcl.2018.02.048","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2018.02.048","pmid":"29519738","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/29519738\/","year":2018,"journal":"Bioorg Med Chem Lett","volume":"28","issue":"7","page":"1211-1218","authors":[{"first_name":"Behera D","last_name":null,"full_name":null},{"first_name":"Deshmukh S","last_name":null,"full_name":null},{"first_name":"Gharat LA.","last_name":null,"full_name":null},{"first_name":"Gudi GS","last_name":null,"full_name":null},{"first_name":"Honnegowda S","last_name":null,"full_name":null},{"first_name":"Jadhav SB","last_name":null,"full_name":null},{"first_name":"Karande V","last_name":null,"full_name":null},{"first_name":"Kattige VG","last_name":null,"full_name":null},{"first_name":"Khairatkar-Joshi N","last_name":null,"full_name":null},{"first_name":"Kulkarni A","last_name":null,"full_name":null},{"first_name":"Muthukaman N","last_name":null,"full_name":null},{"first_name":"Pisal D","last_name":null,"full_name":null},{"first_name":"Pisat M","last_name":null,"full_name":null},{"first_name":"Sangana RR","last_name":null,"full_name":null},{"first_name":"Sarode N","last_name":null,"full_name":null},{"first_name":"Sawant P","last_name":null,"full_name":null},{"first_name":"Shaikh M","last_name":null,"full_name":null},{"first_name":"Tambe M","last_name":null,"full_name":null},{"first_name":"Tondlekar S","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2739","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2739","created_at":"2023-06-23T15:09:32.000000Z","updated_at":null}}