{"data":{"id":2668,"citation":"Verhoest PR, Basak AS, Parikh V, Hayward M, Kauffman GW, Paradis V, McHardy SF, McLean S, Grimwood S, Schmidt AW, Vanase-Frawley M, Freeman J, Van Deusen J, Cox L, Wong D, Liras S.: Design and discovery of a selective small molecule \u03ba opioid antagonist (2-methyl-N-((2'-(pyrrolidin-1-ylsulfonyl)biphenyl-4-yl)methyl)propan-1-amine, PF-4455242). J Med Chem, Volume 54 (16), 2011","title":"Design and discovery of a selective small molecule \u03ba opioid antagonist (2-methyl-N-((2'-(pyrrolidin-1-ylsulfonyl)biphenyl-4-yl)methyl)propan-1-amine, PF-4455242).","doi":"10.1021\/jm2006035","doi_url":"https:\/\/doi.org\/10.1021\/jm2006035","pmid":"21744827","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/21744827\/","year":2011,"journal":"J Med Chem","volume":"54","issue":"16","page":"5868-5877","authors":[{"first_name":"Basak AS","last_name":null,"full_name":null},{"first_name":"Cox L","last_name":null,"full_name":null},{"first_name":"Freeman J","last_name":null,"full_name":null},{"first_name":"Grimwood S","last_name":null,"full_name":null},{"first_name":"Hayward M","last_name":null,"full_name":null},{"first_name":"Kauffman GW","last_name":null,"full_name":null},{"first_name":"Liras S.","last_name":null,"full_name":null},{"first_name":"McHardy SF","last_name":null,"full_name":null},{"first_name":"McLean S","last_name":null,"full_name":null},{"first_name":"Paradis V","last_name":null,"full_name":null},{"first_name":"Parikh V","last_name":null,"full_name":null},{"first_name":"Schmidt AW","last_name":null,"full_name":null},{"first_name":"Van Deusen J","last_name":null,"full_name":null},{"first_name":"Vanase-Frawley M","last_name":null,"full_name":null},{"first_name":"Verhoest PR","last_name":null,"full_name":null},{"first_name":"Wong D","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2668","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2668","created_at":"2023-06-23T15:09:15.000000Z","updated_at":null}}