{"data":{"id":2657,"citation":"Anselm L, Banner DW, Benz J, Zbinden KG, Himber J, Hilpert H, Huber W, Kuhn B, Mary JL, Otteneder MB, Panday N, Ricklin F, Stahl M, Thomi S, Haap W.: Discovery of a factor Xa inhibitor (3R,4R)-1-(2,2-difluoro-ethyl)-pyrrolidine-3,4-dicarboxylic acid 3-[(5-chloro-pyridin-2-yl)-amide] 4-[[2-fluoro-4-(2-oxo-2H-pyridin-1-yl)-phenyl]-amide] as a clinical candidate. Bioorg Med Chem Lett, Volume 20 (17), 2010","title":"Discovery of a factor Xa inhibitor (3R,4R)-1-(2,2-difluoro-ethyl)-pyrrolidine-3,4-dicarboxylic acid 3-[(5-chloro-pyridin-2-yl)-amide] 4-[[2-fluoro-4-(2-oxo-2H-pyridin-1-yl)-phenyl]-amide] as a clinical candidate.","doi":"10.1016\/j.bmcl.2010.06.126","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2010.06.126","pmid":"20650636","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20650636\/","year":2010,"journal":"Bioorg Med Chem Lett","volume":"20","issue":"17","page":"5313-5319","authors":[{"first_name":"Anselm L","last_name":null,"full_name":null},{"first_name":"Banner DW","last_name":null,"full_name":null},{"first_name":"Benz J","last_name":null,"full_name":null},{"first_name":"Haap W.","last_name":null,"full_name":null},{"first_name":"Hilpert H","last_name":null,"full_name":null},{"first_name":"Himber J","last_name":null,"full_name":null},{"first_name":"Huber W","last_name":null,"full_name":null},{"first_name":"Kuhn B","last_name":null,"full_name":null},{"first_name":"Mary JL","last_name":null,"full_name":null},{"first_name":"Otteneder MB","last_name":null,"full_name":null},{"first_name":"Panday N","last_name":null,"full_name":null},{"first_name":"Ricklin F","last_name":null,"full_name":null},{"first_name":"Stahl M","last_name":null,"full_name":null},{"first_name":"Thomi S","last_name":null,"full_name":null},{"first_name":"Zbinden KG","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2657","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2657","created_at":"2023-06-23T15:09:13.000000Z","updated_at":null}}