{"data":{"id":2641,"citation":"Achermann G, Ballard TM, Blasco F, Broutin PE, B\u00fcttelmann B, Fischer H, Graf M, Hernandez MC, Hilty P, Knoflach F, Koblet A, Knust H, Kurt A, Martin JR, Masciadri R, Porter RH, Stadler H, Thomas AW, Trube G, Wichmann J.: Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA(A) alpha5 inverse agonist series. Bioorg Med Chem Lett, Volume 19 (19), 2009","title":"Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA(A) alpha5 inverse agonist series.","doi":"10.1016\/j.bmcl.2009.07.153","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2009.07.153","pmid":"19726184","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/19726184\/","year":2009,"journal":"Bioorg Med Chem Lett","volume":"19","issue":"19","page":"5746-5752","authors":[{"first_name":"Achermann G","last_name":null,"full_name":null},{"first_name":"Ballard TM","last_name":null,"full_name":null},{"first_name":"Blasco F","last_name":null,"full_name":null},{"first_name":"Broutin PE","last_name":null,"full_name":null},{"first_name":"B\u00fcttelmann B","last_name":null,"full_name":null},{"first_name":"Fischer H","last_name":null,"full_name":null},{"first_name":"Graf M","last_name":null,"full_name":null},{"first_name":"Hernandez MC","last_name":null,"full_name":null},{"first_name":"Hilty P","last_name":null,"full_name":null},{"first_name":"Knoflach F","last_name":null,"full_name":null},{"first_name":"Knust H","last_name":null,"full_name":null},{"first_name":"Koblet A","last_name":null,"full_name":null},{"first_name":"Kurt A","last_name":null,"full_name":null},{"first_name":"Martin JR","last_name":null,"full_name":null},{"first_name":"Masciadri R","last_name":null,"full_name":null},{"first_name":"Porter RH","last_name":null,"full_name":null},{"first_name":"Stadler H","last_name":null,"full_name":null},{"first_name":"Thomas AW","last_name":null,"full_name":null},{"first_name":"Trube G","last_name":null,"full_name":null},{"first_name":"Wichmann J.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2641","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2641","created_at":"2023-06-23T15:09:09.000000Z","updated_at":null}}