{"data":{"id":2601,"citation":"Carcache DA, Vulpetti A, Kallen J, Mattes H, Orain D, Stringer R, Vangrevelinghe E, Wolf RM, Kaupmann K, Ottl J, Dawson J, Cooke NG, Hoegenauer K, Billich A, Wagner J, Guntermann C, Hintermann S.: Optimizing a Weakly Binding Fragment into a Potent ROR\u03b3t Inverse Agonist with Efficacy in an in Vivo Inflammation Model. J Med Chem, Volume 61 (15), 2018","title":"Optimizing a Weakly Binding Fragment into a Potent ROR\u03b3t Inverse Agonist with Efficacy in an in Vivo Inflammation Model.","doi":"10.1021\/acs.jmedchem.8b00529","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.8b00529","pmid":"29990434","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/29990434\/","year":2018,"journal":"J Med Chem","volume":"61","issue":"15","page":"6724-6735","authors":[{"first_name":"Billich A","last_name":null,"full_name":null},{"first_name":"Carcache DA","last_name":null,"full_name":null},{"first_name":"Cooke NG","last_name":null,"full_name":null},{"first_name":"Dawson J","last_name":null,"full_name":null},{"first_name":"Guntermann C","last_name":null,"full_name":null},{"first_name":"Hintermann S.","last_name":null,"full_name":null},{"first_name":"Hoegenauer K","last_name":null,"full_name":null},{"first_name":"Kallen J","last_name":null,"full_name":null},{"first_name":"Kaupmann K","last_name":null,"full_name":null},{"first_name":"Mattes H","last_name":null,"full_name":null},{"first_name":"Orain D","last_name":null,"full_name":null},{"first_name":"Ottl J","last_name":null,"full_name":null},{"first_name":"Stringer R","last_name":null,"full_name":null},{"first_name":"Vangrevelinghe E","last_name":null,"full_name":null},{"first_name":"Vulpetti A","last_name":null,"full_name":null},{"first_name":"Wagner J","last_name":null,"full_name":null},{"first_name":"Wolf RM","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2601","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2601","created_at":"2023-06-23T15:09:00.000000Z","updated_at":null}}