{"data":{"id":2588,"citation":"Holzer P, Masuya K, Furet P, Kallen J, Valat-Stachyra T, Ferretti S, Berghausen J, Bouisset-Leonard M, Buschmann N, Pissot-Soldermann C, Rynn C, Ruetz S, Stutz S, Ch\u00e8ne P, Jeay S, Gessier F.: Discovery of a Dihydroisoquinolinone Derivative (NVP-CGM097): A Highly Potent and Selective MDM2 Inhibitor Undergoing Phase 1 Clinical Trials in p53wt Tumors. J Med Chem, Volume 58 (16), 2015","title":"Discovery of a Dihydroisoquinolinone Derivative (NVP-CGM097): A Highly Potent and Selective MDM2 Inhibitor Undergoing Phase 1 Clinical Trials in p53wt Tumors.","doi":"10.1021\/acs.jmedchem.5b00810","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.5b00810","pmid":"26181851","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/26181851\/","year":2015,"journal":"J Med Chem","volume":"58","issue":"16","page":"6348-6358","authors":[{"first_name":"Berghausen J","last_name":null,"full_name":null},{"first_name":"Bouisset-Leonard M","last_name":null,"full_name":null},{"first_name":"Buschmann N","last_name":null,"full_name":null},{"first_name":"Ch\u00e8ne P","last_name":null,"full_name":null},{"first_name":"Ferretti S","last_name":null,"full_name":null},{"first_name":"Furet P","last_name":null,"full_name":null},{"first_name":"Gessier F.","last_name":null,"full_name":null},{"first_name":"Holzer P","last_name":null,"full_name":null},{"first_name":"Jeay S","last_name":null,"full_name":null},{"first_name":"Kallen J","last_name":null,"full_name":null},{"first_name":"Masuya K","last_name":null,"full_name":null},{"first_name":"Pissot-Soldermann C","last_name":null,"full_name":null},{"first_name":"Ruetz S","last_name":null,"full_name":null},{"first_name":"Rynn C","last_name":null,"full_name":null},{"first_name":"Stutz S","last_name":null,"full_name":null},{"first_name":"Valat-Stachyra T","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2588","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2588","created_at":"2023-06-23T15:08:57.000000Z","updated_at":null}}