{"data":{"id":2544,"citation":"Asano T, Yamazaki H, Kasahara C, Kubota H, Kontani T, Harayama Y, Ohno K, Mizuhara H, Yokomoto M, Misumi K, Kinoshita T, Ohta M, Takeuchi M.: Identification, synthesis, and biological evaluation of 6-[(6R)-2-(4-fluorophenyl)-6-(hydroxymethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-2-(2-methylphenyl)pyridazin-3(2H)-one (AS1940477), a potent p38 MAP kinase inhibitor. J Med Chem, Volume 55 (17), 2012","title":"Identification, synthesis, and biological evaluation of 6-[(6R)-2-(4-fluorophenyl)-6-(hydroxymethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-2-(2-methylphenyl)pyridazin-3(2H)-one (AS1940477), a potent p38 MAP kinase inhibitor.","doi":"10.1021\/jm3008008","doi_url":"https:\/\/doi.org\/10.1021\/jm3008008","pmid":"22905713","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/22905713\/","year":2012,"journal":"J Med Chem","volume":"55","issue":"17","page":"7772-7785","authors":[{"first_name":"Asano T","last_name":null,"full_name":null},{"first_name":"Harayama Y","last_name":null,"full_name":null},{"first_name":"Kasahara C","last_name":null,"full_name":null},{"first_name":"Kinoshita T","last_name":null,"full_name":null},{"first_name":"Kontani T","last_name":null,"full_name":null},{"first_name":"Kubota H","last_name":null,"full_name":null},{"first_name":"Misumi K","last_name":null,"full_name":null},{"first_name":"Mizuhara H","last_name":null,"full_name":null},{"first_name":"Ohno K","last_name":null,"full_name":null},{"first_name":"Ohta M","last_name":null,"full_name":null},{"first_name":"Takeuchi M.","last_name":null,"full_name":null},{"first_name":"Yamazaki H","last_name":null,"full_name":null},{"first_name":"Yokomoto M","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2544","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2544","created_at":"2023-06-23T15:08:46.000000Z","updated_at":null}}