{"data":{"id":2459,"citation":"Naud S, Westwood IM, Faisal A, Sheldrake P, Bavetsias V, Atrash B, Cheung KM, Liu M, Hayes A, Schmitt J, Wood A, Choi V, Boxall K, Mak G, Gurden M, Valenti M, de Haven Brandon A, Henley A, Baker R, McAndrew C, Matijssen B, Burke R, Hoelder S, Eccles SA, Raynaud FI, Linardopoulos S, van Montfort RL, Blagg J.: Structure-based design of orally bioavailable 1H-pyrrolo[3,2-c]pyridine inhibitors of mitotic kinase monopolar spindle 1 (MPS1). J Med Chem, Volume 56 (24), 2013","title":"Structure-based design of orally bioavailable 1H-pyrrolo[3,2-c]pyridine inhibitors of mitotic kinase monopolar spindle 1 (MPS1).","doi":"10.1021\/jm401395s","doi_url":"https:\/\/doi.org\/10.1021\/jm401395s","pmid":"24256217","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/24256217\/","year":2013,"journal":"J Med Chem","volume":"56","issue":"24","page":"10045-10065","authors":[{"first_name":"Atrash B","last_name":null,"full_name":null},{"first_name":"Baker R","last_name":null,"full_name":null},{"first_name":"Bavetsias V","last_name":null,"full_name":null},{"first_name":"Blagg J.","last_name":null,"full_name":null},{"first_name":"Boxall K","last_name":null,"full_name":null},{"first_name":"Burke R","last_name":null,"full_name":null},{"first_name":"Cheung KM","last_name":null,"full_name":null},{"first_name":"Choi V","last_name":null,"full_name":null},{"first_name":"de Haven Brandon A","last_name":null,"full_name":null},{"first_name":"Eccles SA","last_name":null,"full_name":null},{"first_name":"Faisal A","last_name":null,"full_name":null},{"first_name":"Gurden M","last_name":null,"full_name":null},{"first_name":"Hayes A","last_name":null,"full_name":null},{"first_name":"Henley A","last_name":null,"full_name":null},{"first_name":"Hoelder S","last_name":null,"full_name":null},{"first_name":"Linardopoulos S","last_name":null,"full_name":null},{"first_name":"Liu M","last_name":null,"full_name":null},{"first_name":"Mak G","last_name":null,"full_name":null},{"first_name":"Matijssen B","last_name":null,"full_name":null},{"first_name":"McAndrew C","last_name":null,"full_name":null},{"first_name":"Naud S","last_name":null,"full_name":null},{"first_name":"Raynaud FI","last_name":null,"full_name":null},{"first_name":"Schmitt J","last_name":null,"full_name":null},{"first_name":"Sheldrake P","last_name":null,"full_name":null},{"first_name":"Valenti M","last_name":null,"full_name":null},{"first_name":"van Montfort RL","last_name":null,"full_name":null},{"first_name":"Westwood IM","last_name":null,"full_name":null},{"first_name":"Wood A","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2459","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2459","created_at":"2023-06-23T15:08:28.000000Z","updated_at":null}}