{"data":{"id":2444,"citation":"Maloney PR, Khan P, Hedrick M, Gosalia P, Milewski M, Li L, Roth GP, Sergienko E, Suyama E, Sugarman E, Nguyen K, Mehta A, Vasile S, Su Y, Stonich D, Nguyen H, Zeng FY, Novo AM, Vicchiarelli M, Diwan J, Chung TD, Smith LH, Pinkerton AB.: Discovery of 4-oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 4-nitrobenzoate (ML221) as a functional antagonist of the apelin (APJ) receptor. Bioorg Med Chem Lett, Volume 22 (21), 2012","title":"Discovery of 4-oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 4-nitrobenzoate (ML221) as a functional antagonist of the apelin (APJ) receptor.","doi":"10.1016\/j.bmcl.2012.08.105","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2012.08.105","pmid":"23010269","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/23010269\/","year":2012,"journal":"Bioorg Med Chem Lett","volume":"22","issue":"21","page":"6656-6660","authors":[{"first_name":"Chung TD","last_name":null,"full_name":null},{"first_name":"Diwan J","last_name":null,"full_name":null},{"first_name":"Gosalia P","last_name":null,"full_name":null},{"first_name":"Hedrick M","last_name":null,"full_name":null},{"first_name":"Khan P","last_name":null,"full_name":null},{"first_name":"Li L","last_name":null,"full_name":null},{"first_name":"Maloney PR","last_name":null,"full_name":null},{"first_name":"Mehta A","last_name":null,"full_name":null},{"first_name":"Milewski M","last_name":null,"full_name":null},{"first_name":"Nguyen H","last_name":null,"full_name":null},{"first_name":"Nguyen K","last_name":null,"full_name":null},{"first_name":"Novo AM","last_name":null,"full_name":null},{"first_name":"Pinkerton AB.","last_name":null,"full_name":null},{"first_name":"Roth GP","last_name":null,"full_name":null},{"first_name":"Sergienko E","last_name":null,"full_name":null},{"first_name":"Smith LH","last_name":null,"full_name":null},{"first_name":"Stonich D","last_name":null,"full_name":null},{"first_name":"Su Y","last_name":null,"full_name":null},{"first_name":"Sugarman E","last_name":null,"full_name":null},{"first_name":"Suyama E","last_name":null,"full_name":null},{"first_name":"Vasile S","last_name":null,"full_name":null},{"first_name":"Vicchiarelli M","last_name":null,"full_name":null},{"first_name":"Zeng FY","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2444","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2444","created_at":"2023-06-23T15:08:25.000000Z","updated_at":null}}