{"data":{"id":2435,"citation":"Engelhardt H, B\u00f6se D, Petronczki M, Scharn D, Bader G, Baum A, Bergner A, Chong E, D\u00f6bel S, Egger G, Engelhardt C, Ettmayer P, Fuchs JE, Gerstberger T, Gonnella N, Grimm A, Grondal E, Haddad N, Hopfgartner B, Kousek R, Krawiec M, Kriz M, Lamarre L, Leung J, Mayer M, Patel ND, Simov BP, Reeves JT, Schnitzer R, Schrenk A, Sharps B, Solca F, Stadtm\u00fcller H, Tan Z, Wunberg T, Zoephel A, McConnell DB.: Start Selective and Rigidify: The Discovery Path toward a Next Generation of EGFR Tyrosine Kinase Inhibitors. J Med Chem, Volume 62 (22), 2019","title":"Start Selective and Rigidify: The Discovery Path toward a Next Generation of EGFR Tyrosine Kinase Inhibitors.","doi":"10.1021\/acs.jmedchem.9b01169","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.9b01169","pmid":"31689114","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/31689114\/","year":2019,"journal":"J Med Chem","volume":"62","issue":"22","page":"10272-10293","authors":[{"first_name":"Bader G","last_name":null,"full_name":null},{"first_name":"Baum A","last_name":null,"full_name":null},{"first_name":"Bergner A","last_name":null,"full_name":null},{"first_name":"B\u00f6se D","last_name":null,"full_name":null},{"first_name":"Chong E","last_name":null,"full_name":null},{"first_name":"D\u00f6bel S","last_name":null,"full_name":null},{"first_name":"Egger G","last_name":null,"full_name":null},{"first_name":"Engelhardt C","last_name":null,"full_name":null},{"first_name":"Engelhardt H","last_name":null,"full_name":null},{"first_name":"Ettmayer P","last_name":null,"full_name":null},{"first_name":"Fuchs JE","last_name":null,"full_name":null},{"first_name":"Gerstberger T","last_name":null,"full_name":null},{"first_name":"Gonnella N","last_name":null,"full_name":null},{"first_name":"Grimm A","last_name":null,"full_name":null},{"first_name":"Grondal E","last_name":null,"full_name":null},{"first_name":"Haddad N","last_name":null,"full_name":null},{"first_name":"Hopfgartner B","last_name":null,"full_name":null},{"first_name":"Kousek R","last_name":null,"full_name":null},{"first_name":"Krawiec M","last_name":null,"full_name":null},{"first_name":"Kriz M","last_name":null,"full_name":null},{"first_name":"Lamarre L","last_name":null,"full_name":null},{"first_name":"Leung J","last_name":null,"full_name":null},{"first_name":"Mayer M","last_name":null,"full_name":null},{"first_name":"McConnell DB.","last_name":null,"full_name":null},{"first_name":"Patel ND","last_name":null,"full_name":null},{"first_name":"Petronczki M","last_name":null,"full_name":null},{"first_name":"Reeves JT","last_name":null,"full_name":null},{"first_name":"Scharn D","last_name":null,"full_name":null},{"first_name":"Schnitzer R","last_name":null,"full_name":null},{"first_name":"Schrenk A","last_name":null,"full_name":null},{"first_name":"Sharps B","last_name":null,"full_name":null},{"first_name":"Simov BP","last_name":null,"full_name":null},{"first_name":"Solca F","last_name":null,"full_name":null},{"first_name":"Stadtm\u00fcller H","last_name":null,"full_name":null},{"first_name":"Tan Z","last_name":null,"full_name":null},{"first_name":"Wunberg T","last_name":null,"full_name":null},{"first_name":"Zoephel A","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2435","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2435","created_at":"2023-06-23T15:08:23.000000Z","updated_at":null}}