{"data":{"id":2284,"citation":"Truong AP, Probst GD, Aquino J, Fang L, Brogley L, Sealy JM, Hom RK, Tucker JA, John V, Tung JS, Pleiss MA, Konradi AW, Sham HL, Dappen MS, T\u00f3th G, Yao N, Brecht E, Pan H, Artis DR, Ruslim L, Bova MP, Sinha S, Yednock TA, Zmolek W, Quinn KP, Sauer JM.: Improving the permeability of the hydroxyethylamine BACE-1 inhibitors: structure-activity relationship of P2' substituents. Bioorg Med Chem Lett, Volume 20 (16), 2010","title":"Improving the permeability of the hydroxyethylamine BACE-1 inhibitors: structure-activity relationship of P2' substituents.","doi":"10.1016\/j.bmcl.2010.06.112","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2010.06.112","pmid":"20634069","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20634069\/","year":2010,"journal":"Bioorg Med Chem Lett","volume":"20","issue":"16","page":"4789-4794","authors":[{"first_name":"Aquino J","last_name":null,"full_name":null},{"first_name":"Artis DR","last_name":null,"full_name":null},{"first_name":"Bova MP","last_name":null,"full_name":null},{"first_name":"Brecht E","last_name":null,"full_name":null},{"first_name":"Brogley L","last_name":null,"full_name":null},{"first_name":"Dappen MS","last_name":null,"full_name":null},{"first_name":"Fang L","last_name":null,"full_name":null},{"first_name":"Hom RK","last_name":null,"full_name":null},{"first_name":"John V","last_name":null,"full_name":null},{"first_name":"Konradi AW","last_name":null,"full_name":null},{"first_name":"Pan H","last_name":null,"full_name":null},{"first_name":"Pleiss MA","last_name":null,"full_name":null},{"first_name":"Probst GD","last_name":null,"full_name":null},{"first_name":"Quinn KP","last_name":null,"full_name":null},{"first_name":"Ruslim L","last_name":null,"full_name":null},{"first_name":"Sealy JM","last_name":null,"full_name":null},{"first_name":"Sham HL","last_name":null,"full_name":null},{"first_name":"Sinha S","last_name":null,"full_name":null},{"first_name":"Toth G","last_name":null,"full_name":null},{"first_name":"Truong AP","last_name":null,"full_name":null},{"first_name":"Tucker JA","last_name":null,"full_name":null},{"first_name":"Tung JS","last_name":null,"full_name":null},{"first_name":"Yao N","last_name":null,"full_name":null},{"first_name":"Yednock TA","last_name":null,"full_name":null},{"first_name":"Zmolek W","last_name":null,"full_name":null},{"first_name":"Sauer JM.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2284","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2284","created_at":"2023-06-23T10:46:16.000000Z","updated_at":null}}