{"data":{"id":2221,"citation":"Wittman MD, Carboni JM, Yang Z, Lee FY, Antman M, Attar R, Balimane P, Chang C, Chen C, Discenza L, Frennesson D, Gottardis MM, Greer A, Hurlburt W, Johnson W, Langley DR, Li A, Li J, Liu P, Mastalerz H, Mathur A, Menard K, Patel K, Sack J, Sang X, Saulnier M, Smith D, Stefanski K, Trainor G, Velaparthi U, Zhang G, Zimmermann K, Vyas DM.: Discovery of a 2,4-disubstituted pyrrolo[1,2-f][1,2,4]triazine inhibitor (BMS-754807) of insulin-like growth factor receptor (IGF-1R) kinase in clinical development. J Med Chem, Volume 52 (23), 2009","title":"Discovery of a 2,4-disubstituted pyrrolo[1,2-f][1,2,4]triazine inhibitor (BMS-754807) of insulin-like growth factor receptor (IGF-1R) kinase in clinical development.","doi":"10.1021\/jm900786r","doi_url":"https:\/\/doi.org\/10.1021\/jm900786r","pmid":"19778024","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/19778024\/","year":2009,"journal":"J Med Chem","volume":"52","issue":"23","page":"7360-7363","authors":[{"first_name":"Antman M","last_name":null,"full_name":null},{"first_name":"Attar R","last_name":null,"full_name":null},{"first_name":"Balimane P","last_name":null,"full_name":null},{"first_name":"Carboni JM","last_name":null,"full_name":null},{"first_name":"Chang C","last_name":null,"full_name":null},{"first_name":"Chen C","last_name":null,"full_name":null},{"first_name":"Discenza L","last_name":null,"full_name":null},{"first_name":"Frennesson D","last_name":null,"full_name":null},{"first_name":"Gottardis MM","last_name":null,"full_name":null},{"first_name":"Greer A","last_name":null,"full_name":null},{"first_name":"Hurlburt W","last_name":null,"full_name":null},{"first_name":"Johnson W","last_name":null,"full_name":null},{"first_name":"Langley DR","last_name":null,"full_name":null},{"first_name":"Lee FY","last_name":null,"full_name":null},{"first_name":"Li A","last_name":null,"full_name":null},{"first_name":"Li J","last_name":null,"full_name":null},{"first_name":"Liu P","last_name":null,"full_name":null},{"first_name":"Mastalerz H","last_name":null,"full_name":null},{"first_name":"Mathur A","last_name":null,"full_name":null},{"first_name":"Menard K","last_name":null,"full_name":null},{"first_name":"Patel K","last_name":null,"full_name":null},{"first_name":"Sack J","last_name":null,"full_name":null},{"first_name":"Sang X","last_name":null,"full_name":null},{"first_name":"Saulnier M","last_name":null,"full_name":null},{"first_name":"Smith D","last_name":null,"full_name":null},{"first_name":"Stefanski K","last_name":null,"full_name":null},{"first_name":"Trainor G","last_name":null,"full_name":null},{"first_name":"Velaparthi U","last_name":null,"full_name":null},{"first_name":"Vyas DM.","last_name":null,"full_name":null},{"first_name":"Wittman MD","last_name":null,"full_name":null},{"first_name":"Yang Z","last_name":null,"full_name":null},{"first_name":"Zhang G","last_name":null,"full_name":null},{"first_name":"Zimmermann K","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2221","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2221","created_at":"2023-06-23T10:10:35.000000Z","updated_at":null}}