{"data":{"id":2079,"citation":"Fattori D, Porcelloni M, D'Andrea P, Catalioto RM, Ettorre A, Giuliani S, Marastoni E, Mauro S, Meini S, Rossi C, Altamura M, Maggi CA.: Structure-activity relationships of 6-methyl-benzo[b]thiophene-2-carboxylic acid (1-[(S)-1-benzyl-4-[4-(tetrahydropyran-4-ylmethyl)piperazin-1-yl]butylcarbamoyl]cyclopentyl)amide, potent antagonist of the neurokinin-2 receptor. J Med Chem, Volume 53 (10), 2010","title":"Structure-activity relationships of 6-methyl-benzo[b]thiophene-2-carboxylic acid (1-[(S)-1-benzyl-4-[4-(tetrahydropyran-4-ylmethyl)piperazin-1-yl]butylcarbamoyl]cyclopentyl)amide, potent antagonist of the neurokinin-2 receptor.","doi":"10.1021\/jm100176s","doi_url":"https:\/\/doi.org\/10.1021\/jm100176s","pmid":"20408549","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20408549\/","year":2010,"journal":"J Med Chem","volume":"53","issue":"10","page":"4148-4165","authors":[{"first_name":"Altamura M","last_name":null,"full_name":null},{"first_name":"Catalioto RM","last_name":null,"full_name":null},{"first_name":"D'Andrea P","last_name":null,"full_name":null},{"first_name":"Ettorre A","last_name":null,"full_name":null},{"first_name":"Fattori D","last_name":null,"full_name":null},{"first_name":"Giuliani S","last_name":null,"full_name":null},{"first_name":"Maggi CA.","last_name":null,"full_name":null},{"first_name":"Marastoni E","last_name":null,"full_name":null},{"first_name":"Mauro S","last_name":null,"full_name":null},{"first_name":"Meini S","last_name":null,"full_name":null},{"first_name":"Porcelloni M","last_name":null,"full_name":null},{"first_name":"Rossi C","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2079","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2079","created_at":"2023-06-23T10:10:03.000000Z","updated_at":null}}