{"data":{"id":2051,"citation":"Lemoine RC, Petersen AC, Setti L, Wanner J, Jekle A, Heilek G, deRosier A, Ji C, Berry P, Rotstein D.: Evaluation of secondary amide replacements in a series of CCR5 antagonists as a means to increase intrinsic membrane permeability. Part 1: Optimization of gem-disubstituted azacycles. Bioorg Med Chem Lett, Volume 20 (2), 2010","title":"Evaluation of secondary amide replacements in a series of CCR5 antagonists as a means to increase intrinsic membrane permeability. Part 1: Optimization of gem-disubstituted azacycles.","doi":"10.1016\/j.bmcl.2009.11.072","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2009.11.072","pmid":"20004099","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20004099\/","year":2010,"journal":"Bioorg Med Chem Lett","volume":"20","issue":"2","page":"704-708","authors":[{"first_name":"Berry P","last_name":null,"full_name":null},{"first_name":"deRosier A","last_name":null,"full_name":null},{"first_name":"Heilek G","last_name":null,"full_name":null},{"first_name":"Jekle A","last_name":null,"full_name":null},{"first_name":"Ji C","last_name":null,"full_name":null},{"first_name":"Lemoine RC","last_name":null,"full_name":null},{"first_name":"Petersen AC","last_name":null,"full_name":null},{"first_name":"Rotstein D.","last_name":null,"full_name":null},{"first_name":"Setti L","last_name":null,"full_name":null},{"first_name":"Wanner J","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2051","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2051","created_at":"2023-06-23T10:09:58.000000Z","updated_at":null}}