{"data":{"id":1476,"citation":"Czodrowski P, Mallinger A, Wienke D, Esdar C, P\u00f6schke O, Busch M, Rohdich F, Eccles SA, Ortiz-Ruiz MJ, Schneider R, Raynaud FI, Clarke PA, Musil D, Schwarz D, Dale T, Urbahns K, Blagg J, Schiemann K.: Structure-Based Optimization of Potent, Selective, and Orally Bioavailable CDK8 Inhibitors Discovered by High-Throughput Screening. J Med Chem, Volume 59 (20), 2016","title":"Structure-Based Optimization of Potent, Selective, and Orally Bioavailable CDK8 Inhibitors Discovered by High-Throughput Screening.","doi":"10.1021\/acs.jmedchem.6b00597","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.6b00597","pmid":"27490956","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/27490956\/","year":2016,"journal":"J Med Chem","volume":"59","issue":"20","page":"9337-9349","authors":[{"first_name":"Blagg J","last_name":null,"full_name":null},{"first_name":"Busch M","last_name":null,"full_name":null},{"first_name":"Clarke PA","last_name":null,"full_name":null},{"first_name":"Czodrowski P","last_name":null,"full_name":null},{"first_name":"Dale T","last_name":null,"full_name":null},{"first_name":"Eccles SA","last_name":null,"full_name":null},{"first_name":"Esdar C","last_name":null,"full_name":null},{"first_name":"Mallinger A","last_name":null,"full_name":null},{"first_name":"Musil D","last_name":null,"full_name":null},{"first_name":"Ortiz-Ruiz MJ","last_name":null,"full_name":null},{"first_name":"P\u00f6schke O","last_name":null,"full_name":null},{"first_name":"Raynaud FI","last_name":null,"full_name":null},{"first_name":"Rohdich F","last_name":null,"full_name":null},{"first_name":"Schiemann K.","last_name":null,"full_name":null},{"first_name":"Schneider R","last_name":null,"full_name":null},{"first_name":"Schwarz D","last_name":null,"full_name":null},{"first_name":"Urbahns K","last_name":null,"full_name":null},{"first_name":"Wienke D","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/1476","landing_page":"https:\/\/molmedb.upol.cz\/publication\/1476","created_at":"2021-01-20T12:16:51.000000Z","updated_at":null}}