{"data":{"id":1237,"citation":"Crosignani S, Bingham P, Bottemanne P, Cannelle H, Cauwenberghs S, Cordonnier M, Dalvie D, Deroose F, Feng JL, Gomes B, Greasley S, Kaiser SE, Kraus M, N\u00e9grerie M, Maegley K, Miller N, Murray BW, Schneider M, Soloweij J, Stewart AE, Tumang J, Torti VR, Van Den Eynde B, Wythes M.: Discovery of a Novel and Selective Indoleamine 2,3-Dioxygenase (IDO-1) Inhibitor 3-(5-Fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione (EOS200271\/PF-06840003) and Its Characterization as a Potential Clinical Candidate. J Med Chem, Volume 60 (23), 2017","title":"Discovery of a Novel and Selective Indoleamine 2,3-Dioxygenase (IDO-1) Inhibitor 3-(5-Fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione (EOS200271\/PF-06840003) and Its Characterization as a Potential Clinical Candidate.","doi":"10.1021\/acs.jmedchem.7b00974","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.7b00974","pmid":"29111717","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/29111717\/","year":2017,"journal":"J Med Chem","volume":"60","issue":"23","page":"9617-9629","authors":[{"first_name":"Bingham P","last_name":null,"full_name":null},{"first_name":"Bottemanne P","last_name":null,"full_name":null},{"first_name":"Cannelle H","last_name":null,"full_name":null},{"first_name":"Cauwenberghs S","last_name":null,"full_name":null},{"first_name":"Cordonnier M","last_name":null,"full_name":null},{"first_name":"Crosignani S","last_name":null,"full_name":null},{"first_name":"Dalvie D","last_name":null,"full_name":null},{"first_name":"Deroose F","last_name":null,"full_name":null},{"first_name":"Feng JL","last_name":null,"full_name":null},{"first_name":"Gomes B","last_name":null,"full_name":null},{"first_name":"Greasley S","last_name":null,"full_name":null},{"first_name":"Kaiser SE","last_name":null,"full_name":null},{"first_name":"Kraus M","last_name":null,"full_name":null},{"first_name":"Maegley K","last_name":null,"full_name":null},{"first_name":"Miller N","last_name":null,"full_name":null},{"first_name":"Murray BW","last_name":null,"full_name":null},{"first_name":"N\u00e9grerie M","last_name":null,"full_name":null},{"first_name":"Schneider M","last_name":null,"full_name":null},{"first_name":"Soloweij J","last_name":null,"full_name":null},{"first_name":"Stewart AE","last_name":null,"full_name":null},{"first_name":"Torti VR","last_name":null,"full_name":null},{"first_name":"Tumang J","last_name":null,"full_name":null},{"first_name":"Van Den Eynde B","last_name":null,"full_name":null},{"first_name":"Wythes M.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/1237","landing_page":"https:\/\/molmedb.upol.cz\/publication\/1237","created_at":"2021-01-20T08:41:05.000000Z","updated_at":null}}