{"data":{"id":1064,"citation":"Hudkins RL, Raddatz R, Tao M, Mathiasen JR, Aimone LD, Becknell NC, Prouty CP, Knutsen LJ, Yazdanian M, Moachon G, Ator MA, Mallamo JP, Marino MJ, Bacon ER, Williams M.: Discovery and characterization of 6-{4-[3-(R)-2-methylpyrrolidin-1-yl)propoxy]phenyl}-2H-pyridazin-3-one (CEP-26401, irdabisant): a potent, selective histamine H3 receptor inverse agonist. J Med Chem, Volume 54 (13), 2011","title":"Discovery and characterization of 6-{4-[3-(R)-2-methylpyrrolidin-1-yl)propoxy]phenyl}-2H-pyridazin-3-one (CEP-26401, irdabisant): a potent, selective histamine H3 receptor inverse agonist.","doi":"10.1021\/jm200401v","doi_url":"https:\/\/doi.org\/10.1021\/jm200401v","pmid":"21634396","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/21634396\/","year":2011,"journal":"J Med Chem","volume":"54","issue":"13","page":"4781-4792","authors":[{"first_name":"Aimone LD","last_name":null,"full_name":null},{"first_name":"Ator MA","last_name":null,"full_name":null},{"first_name":"Bacon ER","last_name":null,"full_name":null},{"first_name":"Becknell NC","last_name":null,"full_name":null},{"first_name":"Hudkins RL","last_name":null,"full_name":null},{"first_name":"Knutsen LJ","last_name":null,"full_name":null},{"first_name":"Mallamo JP","last_name":null,"full_name":null},{"first_name":"Marino MJ","last_name":null,"full_name":null},{"first_name":"Mathiasen JR","last_name":null,"full_name":null},{"first_name":"Moachon G","last_name":null,"full_name":null},{"first_name":"Prouty CP","last_name":null,"full_name":null},{"first_name":"Raddatz R","last_name":null,"full_name":null},{"first_name":"Tao M","last_name":null,"full_name":null},{"first_name":"Williams M.","last_name":null,"full_name":null},{"first_name":"Yazdanian M","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/1064","landing_page":"https:\/\/molmedb.upol.cz\/publication\/1064","created_at":"2021-01-20T08:40:10.000000Z","updated_at":null}}